SCHEMBL9753655

SCHEMBL9753655

O=C/C=C/c1c(-c2ccc(F)cc2)nn2cccc2c1C1CC1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 4/20 0.40
ADORA2A P29274 3/20 0.40
ADORA2B P29275 3/20 0.40
ADORA3 P0DMS8 2/20 0.40
ADORA1 P30542 2/20 0.40
EGFR P00533 1/20 0.40
RAF1 P04049 1/20 0.40
GSK3B P49841 1/20 0.40
SLC34A1 Q06495 4/20 0.35
RXRA P19793 1/20 0.35
PTGS2 P35354 2/20 0.34
PTGS1 P23219 2/20 0.33
KDM5B Q9UGL1 1/20 0.32
ALDH1A1 P00352 1/20 0.32
POLB P06746 1/20 0.32
ALOX5 P09917 1/20 0.31
KCNQ3 O43525 1/20 0.31
KCNQ2 O43526 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9753659 1.00 MAPK14 (0.40) MAPK14ADORA2AADORA2BADORA3ADORA1
SCHEMBL9753398 0.89 MAPK14 (0.43) MAPK14ADORA2AADORA2BADORA3ADORA1
SCHEMBL9753011 0.81 MAPK14 (0.43) MAPK14ADORA2AADORA2BADORA3ADORA1
SCHEMBL9753013 0.81 MAPK14 (0.43) MAPK14ADORA2AADORA2BADORA3ADORA1
SCHEMBL9753678 0.79 MAPK14 (0.41) MAPK14ADORA2AADORA2BADORA3ADORA1
SCHEMBL9753675 0.79 MAPK14 (0.41) MAPK14ADORA2AADORA2BADORA3ADORA1
SCHEMBL9753160 0.79 MAPK14 (0.41) MAPK14ADORA2AADORA2BADORA3ADORA1
SCHEMBL9753157 0.79 MAPK14 (0.41) MAPK14ADORA2AADORA2BADORA3ADORA1
SCHEMBL9753303 0.76 PDE4D (0.57) ADORA3RXRAPTGS2ALDH1A1
SCHEMBL9752940 0.74 MAPK14 (0.43) MAPK14ADORA2AADORA2BADORA3ADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991018903-A1 PYRROLOPYRIDAZINE COMPOUNDS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1991-12-12 WO disclosed