SCHEMBL9752940

SCHEMBL9752940

OCc1c(-c2ccc(F)cc2)nn2cccc2c1C1CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 5/20 0.43
EGFR P00533 1/20 0.43
RAF1 P04049 1/20 0.43
ADORA3 P0DMS8 1/20 0.43
ADORA2A P29274 1/20 0.43
ADORA2B P29275 1/20 0.43
ADORA1 P30542 1/20 0.43
GSK3B P49841 1/20 0.43
PRKAA2 P54646 1/20 0.41
SLC34A1 Q06495 4/20 0.36
PTGS1 P23219 1/20 0.35
PTGS2 P35354 1/20 0.35
JAK2 O60674 2/20 0.34
JAK3 P52333 2/20 0.34
PTK2 Q05397 2/20 0.34
KCNQ3 O43525 2/20 0.33
KCNQ2 O43526 2/20 0.33
ALOX5 P09917 1/20 0.33
IDO1 P14902 1/20 0.32
TDO2 P48775 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9753402 0.79 MAPK14 (0.46) MAPK14EGFRRAF1ADORA3ADORA2A
SCHEMBL9753398 0.78 MAPK14 (0.43) MAPK14EGFRRAF1ADORA3ADORA2A
SCHEMBL9753170 0.77 MAPK14 (0.44) MAPK14EGFRRAF1ADORA3ADORA2A
SCHEMBL9753641 0.76 LMNA (0.42) MAPK14EGFRRAF1ADORA3ADORA2A
SCHEMBL9753659 0.74 MAPK14 (0.40) MAPK14EGFRRAF1ADORA3ADORA2A
SCHEMBL9753655 0.74 MAPK14 (0.40) MAPK14EGFRRAF1ADORA3ADORA2A
SCHEMBL9753303 0.70 PDE4D (0.57) ADORA3PTGS2
SCHEMBL3825789 0.69 MAPK14 (0.47) MAPK14EGFRRAF1ADORA3ADORA2A
SCHEMBL10500565 0.67 MAPK14 (0.61) MAPK14EGFRRAF1ADORA3ADORA2A
SCHEMBL14810787 0.67 CYP11B2 (0.47) MAPK14EGFRRAF1ADORA3ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991018903-A1 PYRROLOPYRIDAZINE COMPOUNDS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1991-12-12 WO disclosed
CN-1056690-A PYRROLOPYRIDAZINE COMPOUNDS FUJISAWA PHARMACEUTICAL CO (JP) 1991-12-04 CN disclosed