SCHEMBL9754820

SCHEMBL9754820

CCCc1nc2c(C)cc(C#N)cc2[nH]1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.37
MEN1 O00255 2/20 0.37
ALDH1A1 P00352 3/20 0.36
POLB P06746 2/20 0.36
MAPK1 P28482 1/20 0.36
KDM4E B2RXH2 3/20 0.35
ACACB O00763 1/20 0.34
ACACA Q13085 1/20 0.34
HPGD P15428 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
GRIN1 Q05586 1/20 0.33
GRIN2B Q13224 1/20 0.33
CTSK P43235 3/20 0.33
CSNK1A1 P48729 1/20 0.33
CSNK1D P48730 1/20 0.33
GSK3B P49841 1/20 0.33
CSNK1G2 P78368 1/20 0.33
CYP1A2 P05177 1/20 0.32
GAA P10253 1/20 0.32
CYP2D6 P10635 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19342748 0.83 KDM4E (0.44) KMT2AMEN1ALDH1A1POLBKDM4E
SCHEMBL1918148 0.77 EGLN1 (0.40) KMT2AALDH1A1POLBKDM4EACACB
SCHEMBL9754821 0.77 ADORA1 (0.36) KMT2AMEN1ALDH1A1POLBMAPK1
SCHEMBL14855819 0.75 KMT2A (0.35) KMT2AALDH1A1POLBKDM4EACACB
SCHEMBL3640946 0.75 ACACB (0.36) KMT2AALDH1A1POLBKDM4EACACB
SCHEMBL3712698 0.73 KMT2A (0.38) KMT2AALDH1A1POLBMAPK1KDM4E
SCHEMBL17801869 0.73 KDM4E (0.38) KMT2AALDH1A1POLBKDM4EACACB
SCHEMBL4553606 0.73 ACACB (0.36) KMT2AALDH1A1POLBKDM4EACACB
Hydrochloric Acid SCHEMBL4437775 0.73 ACACB (0.44) KMT2AALDH1A1MAPK1KDM4EACACB
SCHEMBL27809455 0.73 KMT2A (0.36) KMT2APOLBMAPK1KDM4EACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991013063-A1 NEW BENZIMIDAZOLE DERIVATIVES, METHOD FOR PREPARING THEM AND THEIR PHARMACEUTICAL USE SCHERING AKTIENGESELLSCHAFT BERLIN UND BERGKAMEN (DE) 1991-09-05 WO disclosed