SCHEMBL9756716

SCHEMBL9756716

Oc1ccc2c(c1)[CH]NCC2

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 7/20 0.46
DRD4 P21917 2/20 0.46
DRD1 P21728 5/20 0.43
DRD3 P35462 3/20 0.39
DRD5 P21918 2/20 0.39
PBRM1 Q86U86 1/20 0.37
ADCY6 O43306 1/20 0.34
ADCY3 O60266 1/20 0.34
ADCY9 O60503 1/20 0.34
ADCY5 O95622 1/20 0.34
ADCY8 P40145 1/20 0.34
ADCY7 P51828 1/20 0.34
ADCY2 Q08462 1/20 0.34
ADCY1 Q08828 1/20 0.34
ADCY4 Q8NFM4 1/20 0.34
OPRK1 P41145 1/20 0.34
KDM1A O60341 1/20 0.34
CA2 P00918 1/20 0.33
CA5A P35218 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5844893 0.84 DRD2 (0.50) DRD2DRD4DRD1DRD3DRD5
SCHEMBL20520367 0.76 PARP10 (0.44) KDM1A
SCHEMBL19579719 0.70 HTR2C (0.48)
SCHEMBL9618452 0.69
SCHEMBL9529812 0.69 DRD2 (0.47) DRD2DRD4DRD1DRD3DRD5
SCHEMBL7469508 0.68 CA2 (0.43) DRD2DRD4DRD1DRD3DRD5
SCHEMBL4030395 0.68 DRD2 (0.79) DRD2DRD4DRD1DRD3DRD5
SCHEMBL31317940 0.68 DRD2 (0.79) DRD2DRD4DRD1DRD3DRD5
SCHEMBL222933 0.68 HTR2C (0.37) KDM1A
SCHEMBL33917 0.67 DRD2 (0.70) DRD2DRD4DRD1DRD3DRD5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992000072-A1 TETRAHYDROISOQUINOLINYLCARBAMATES OF 1,2,3,3A,8,8A-HEXAHYDRO-1,3A,8-TRIMETHYLPYRROLO[2,3-B]INDOLE HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-01-09 WO disclosed