SCHEMBL9757128

SCHEMBL9757128

N#Cc1nc2ccc(O)cc2o1

nearest known ligand 0.65

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PSMB8 P28062 3/20 0.65
PSMB5 P28074 1/20 0.65
ESR1 P03372 12/20 0.53
ESR2 Q92731 12/20 0.53
APP P05067 1/20 0.46
MIF P14174 1/20 0.45
CA9 Q16790 1/20 0.45
CYP19A1 P11511 1/20 0.44
STS P08842 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9757252 0.79 PSMB8 (0.65) PSMB8PSMB5NPC1RAB9A
SCHEMBL21689039 0.79 PSMB8 (0.65) PSMB8PSMB5APPNPC1RAB9A
SCHEMBL9797527 0.78 PSMB8 (0.63) PSMB8PSMB5
SCHEMBL9797235 0.77 PSMB8 (0.61) PSMB8PSMB5
SCHEMBL17265862 0.75 ESR1 (0.61) ESR1ESR2APPCA9STS
SCHEMBL29999385 0.75 ESR1 (0.61) ESR1ESR2APPCA9STS
SCHEMBL9757041 0.75 PSMB8 (0.59) PSMB8PSMB5CYP19A1NPC1RAB9A
SCHEMBL8740097 0.74 ESR1 (0.74) ESR1ESR2APPCYP19A1NPC1
SCHEMBL27837395 0.74 ESR1 (0.56) ESR1ESR2APPCA9STS
SCHEMBL548913 0.73 PSMB8 (1.00) PSMB8PSMB5NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991019475-A2 QUINOLINYL-BENZOHETEROBICYCLIC DERIVATIVES AS ANTAGONISTS OF LEUKOTRIENE D¿4? RHONE-POULENC RORER INTERNATIONAL (HOLDINGS) INC. (US) 1991-12-26 WO disclosed
US-5041453-A Quinolinyl-benzoheterobicyclic derivatives as antagonists of leukotriene D4 RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1991-08-20 US disclosed