SCHEMBL9757152

SCHEMBL9757152

COC(=O)Cc1nc2ccc(C)cc2o1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.60
KDM4E B2RXH2 2/20 0.60
NPC1 O15118 6/20 0.52
RAB9A P51151 6/20 0.52
SMN1; SMN2 Q16637 3/20 0.52
HSD17B10 Q99714 2/20 0.52
ALDH1A1 P00352 1/20 0.52
HPGD P15428 1/20 0.52
NFKB1 P19838 1/20 0.52
NFKB2 Q00653 1/20 0.52
RELA Q04206 1/20 0.52
ATM Q13315 1/20 0.52
USP2 O75604 1/20 0.50
MAPK10 P53779 1/20 0.50
TP53 P04637 2/20 0.49
AGPAT2 O15120 1/20 0.46
POLB P06746 1/20 0.44
LMNA P02545 1/20 0.44
CACNA1G O43497 1/20 0.43
KCNH2 Q12809 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11333951 0.89 AGPAT2 (0.47) MAPTKDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL10033451 0.86 MAPT (0.66) MAPTKDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL22629662 0.84 NPC1 (0.52) MAPTKDM4ENPC1RAB9ATP53
SCHEMBL11191233 0.84 MAPT (0.66) MAPTKDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL9757094 0.82 NPC1 (0.45) MAPTKDM4ENPC1RAB9AALDH1A1
SCHEMBL5624696 0.81 MAPT (0.54) MAPTKDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL11326015 0.80 RPS6KB2 (0.48) MAPTKDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL14045318 0.76 NPC1 (0.60) MAPTKDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL24766804 0.76 GAA (0.49) MAPTKDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL11310133 0.76 MEN1 (0.55) MAPTKDM4ENPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991019475-A2 QUINOLINYL-BENZOHETEROBICYCLIC DERIVATIVES AS ANTAGONISTS OF LEUKOTRIENE D¿4? RHONE-POULENC RORER INTERNATIONAL (HOLDINGS) INC. (US) 1991-12-26 WO disclosed
US-5041453-A Quinolinyl-benzoheterobicyclic derivatives as antagonists of leukotriene D4 RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1991-08-20 US disclosed