SCHEMBL9763511

SCHEMBL9763511

CSc1ccc(CCCCOCCCCCCBr)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
THRA P10827 1/20 0.38
THRB P10828 1/20 0.38
GAA P10253 1/20 0.37
MEN1 O00255 1/20 0.36
USP2 O75604 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
CYP3A4 P08684 1/20 0.36
MAPK1 P28482 1/20 0.36
CASP1 P29466 1/20 0.36
KMT2A Q03164 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
SLCO1B3 Q9NPD5 1/20 0.36
SLCO1B1 Q9Y6L6 1/20 0.36
SLC6A4 P31645 7/20 0.36
SPHK1 Q9NYA1 1/20 0.35
MAOA P21397 1/20 0.35
SLC6A2 P23975 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10465003 0.97 TDP1 (0.37) TDP1L3MBTL1THRATHRBGAA
SCHEMBL10488711 0.94 KCNH2 (0.37) TDP1L3MBTL1GAASLC6A4MAOA
SCHEMBL7621783 0.90 THRA (0.44) THRATHRBGAAMEN1ALDH1A1
SCHEMBL10867015 0.87 ALDH1A1 (0.35) THRATHRBGAAMEN1USP2
SCHEMBL81028 0.82 SLC6A4 (0.45) GAAMEN1CYP3A4KMT2ASLC6A4
SCHEMBL10465525 0.81 KCNH2 (0.46) TDP1L3MBTL1THRATHRBGAA
SCHEMBL10488103 0.80 TDP1 (0.45) TDP1L3MBTL1THRATHRBMEN1
SCHEMBL9574323 0.79 TDP1 (0.63) TDP1L3MBTL1MEN1USP2ALDH1A1
SCHEMBL9763470 0.78 SLC6A4 (0.38) TDP1L3MBTL1THRATHRBMEN1
SCHEMBL6679345 0.78 TDP1 (0.40) TDP1L3MBTL1THRATHRBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4990505-A Treating asthma, bronchitis; adrenergic stimulants GLAXO GROUP LIMITED (GB) 1991-02-05 US disclosed
US-4853382-A TREATING ASTHMA AND BRONCHITIS GLAXO GROUP LIMITED (GB) 1989-08-01 US disclosed
EP-0178919-B1 AMINOPHENOL DERIVATIVES GLAXO GROUP LIMITED (GB) 1988-12-21 EP disclosed
US-4730008-A STIMULANT FOR BETA-ADRENORECEPTORS GLAXO GROUP LIMITED (GB) 1988-03-08 US disclosed
EP-0178919-A2 Aminophenol derivatives GLAXO GROUP LIMITED (GB) 1986-04-23 EP disclosed