SCHEMBL9763534

SCHEMBL9763534

CC(C)c1c(CBr)n(-c2ccc(F)cc2)c(=O)c2ccccc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.42
ALDH1A1 P00352 2/20 0.42
TDP1 Q9NUW8 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
METAP2 P50579 1/20 0.40
MAPT P10636 2/20 0.39
LMNA P02545 2/20 0.38
PDE10A Q9Y233 1/20 0.38
MAPK1 P28482 1/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
PTGS1 P23219 1/20 0.38
PTGS2 P35354 1/20 0.38
HSD17B10 Q99714 1/20 0.38
CXCR3 P49682 2/20 0.37
PMM2 O15305 1/20 0.37
MPI P34949 1/20 0.37
RAB9A P51151 1/20 0.37
PHOSPHO1 Q8TCT1 1/20 0.37
APOBEC3G Q9HC16 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9763456 0.87 KDM4E (0.44) KDM4EALDH1A1TDP1L3MBTL1METAP2
Bromide SCHEMBL9763504 0.82 KDM4E (0.41) KDM4EALDH1A1TDP1L3MBTL1METAP2
SCHEMBL2676351 0.76 KDM4E (0.48) KDM4EALDH1A1TDP1L3MBTL1METAP2
SCHEMBL9764173 0.76 KDM4E (0.50) KDM4EALDH1A1TDP1L3MBTL1METAP2
SCHEMBL9764267 0.75 KDM4E (0.46) KDM4EALDH1A1TDP1L3MBTL1METAP2
SCHEMBL9763582 0.73 HMGCR (0.49)
SCHEMBL1717723 0.70 TACR3 (0.50) KDM4EALDH1A1LMNAHSD17B10
SCHEMBL9335250 0.70 USP14 (0.38) KDM4EALDH1A1TDP1L3MBTL1
SCHEMBL9763589 0.68 MAPK14 (0.43) KDM4EALDH1A1LMNAPTGS2
SCHEMBL9764024 0.67 HMGCR (0.60) KDM4EALDH1A1LMNAPTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5004747-A Isoquinolinones MAY & BAKER LIMITED (GB) 1991-04-02 US disclosed
EP-0326386-A2 Isoquinolinones MAY & BAKER LIMITED (GB) 1989-08-02 EP disclosed