SCHEMBL9764589

SCHEMBL9764589

O=C(O)/C=C\C(=O)OC(C(=O)O)c1ccccc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 5/20 0.65
ALDH1A1 P00352 2/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
SRC P12931 1/20 0.41
KDM4E B2RXH2 1/20 0.40
MAPT P10636 1/20 0.40
LMNA P02545 2/20 0.39
MAPK1 P28482 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
HDAC3 O15379 1/20 0.38
TNKS O95271 1/20 0.38
HDAC4 P56524 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC7 Q8WUI4 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC10 Q969S8 1/20 0.38
HDAC11 Q96DB2 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
TNKS2 Q9H2K2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11630230 0.83 TDP1 (0.51) HCAR2ALDH1A1CYP2D6MAPTLMNA
SCHEMBL11630234 0.83 TDP1 (0.51) HCAR2ALDH1A1CYP2D6MAPTLMNA
SCHEMBL27534212 0.81 HCAR2 (0.69) HCAR2ALDH1A1CYP2D6SRCKDM4E
SCHEMBL28803484 0.81 HCAR2 (0.69) HCAR2ALDH1A1CYP2D6SRCKDM4E
SCHEMBL7038121 0.81 HCAR2 (0.55) HCAR2ALDH1A1CYP2D6LMNA
SCHEMBL8364617 0.80 CYP2C19 (0.44) HCAR2ALDH1A1CYP3A4CYP2D6SRC
SCHEMBL27722749 0.80 HCAR2 (0.67) HCAR2ALDH1A1CYP2D6KDM4EMAPT
SCHEMBL7086112 0.79 HCAR2 (0.65) HCAR2ALDH1A1CYP3A4CYP2D6SRC
SCHEMBL7089093 0.79 HCAR2 (0.65) HCAR2ALDH1A1CYP3A4CYP2D6SRC
SCHEMBL573378 0.79 HCAR2 (1.00) HCAR2ALDH1A1KDM4EMAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5021413-A Analgesic thiomorpholins their preparation, and pharmaceutical compositions containing them SANKYO COMPANY LIMITED (JP) 1991-06-04 US disclosed