SCHEMBL9765573

SCHEMBL9765573

O=c1c2ccccc2ccc2cc(Cl)c(Cl)cc12

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 2/20 0.47
CYP2A6 P11509 3/20 0.47
PAX8 Q06710 1/20 0.47
CYP1B1 Q16678 3/20 0.46
ALDH1A1 P00352 2/20 0.46
HSD17B10 Q99714 2/20 0.46
HIF1A Q16665 1/20 0.46
CYP1A2 P05177 2/20 0.45
MAPK14 Q16539 2/20 0.44
TSHR P16473 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
GPR84 Q9NQS5 1/20 0.40
CYP1A1 P04798 2/20 0.40
MAPT P10636 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
HPRT1 P00492 1/20 0.39
APAF1 O14727 1/20 0.39
TDP2 O95551 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11723197 0.83 ALDH1A1 (0.48) AKR1B1CYP2A6PAX8CYP1B1ALDH1A1
SCHEMBL9765524 0.82 KDM4E (0.55) AKR1B1CYP2A6PAX8CYP1B1ALDH1A1
SCHEMBL4181934 0.81 ALDH1A1 (0.58) AKR1B1CYP2A6PAX8CYP1B1ALDH1A1
SCHEMBL9212130 0.80 CYP2A6 (0.56) AKR1B1CYP2A6PAX8CYP1B1ALDH1A1
SCHEMBL30186719 0.80 ALDH1A1 (0.65) AKR1B1CYP2A6PAX8CYP1B1ALDH1A1
SCHEMBL268735 0.80 ALDH1A1 (0.65) AKR1B1CYP2A6PAX8CYP1B1ALDH1A1
SCHEMBL29391827 0.80 ALDH1A1 (0.65) AKR1B1CYP2A6PAX8CYP1B1ALDH1A1
SCHEMBL10862574 0.78 CYP1A2 (0.48) AKR1B1CYP2A6CYP1B1ALDH1A1HSD17B10
SCHEMBL9765502 0.76 ALDH1A1 (0.52) AKR1B1CYP2A6PAX8CYP1B1ALDH1A1
SCHEMBL9209062 0.76 CYP2A6 (0.61) AKR1B1CYP2A6PAX8CYP1B1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0272621-B1 Method for the production of 5H-dibenzo[a,d]cyclohepten-5-ones BASF Aktiengesellschaft (DE) 1991-11-27 EP disclosed
US-4845302-A Preparation of 5H-dibenzo[a,d]cyclohepten-5-ones BASF AKTIENGSELLSCHAFT (DE) 1989-07-04 US disclosed
EP-0272621-A2 Method for the production of 5H-dibenzo[a,d]cyclohepten-5-ones BASF Aktiengesellschaft (DE) 1988-06-29 EP disclosed