SCHEMBL9765688

SCHEMBL9765688

COC(=O)C1=C(C)NC(C)=C(C(=O)OC(C)C)C1c1ccccc1C(F)(F)F

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1C Q13936 5/20 0.74
CACNA1F O60840 2/20 0.74
CACNA1D Q01668 2/20 0.74
CACNA1S Q13698 2/20 0.74
CYP1A2 P05177 6/20 0.66
CYP3A4 P08684 6/20 0.66
CYP2C9 P11712 6/20 0.66
CYP2C19 P33261 6/20 0.66
ADORA3 P0DMS8 5/20 0.66
MAPT P10636 4/20 0.66
TSHR P16473 3/20 0.66
NFKB1 P19838 3/20 0.66
CYP2D6 P10635 3/20 0.66
KMT2A Q03164 3/20 0.66
MEN1 O00255 2/20 0.66
NR1I2 O75469 2/20 0.58
ABCB11 O95342 2/20 0.58
KCNH2 Q12809 2/20 0.58
SCN5A Q14524 2/20 0.58
MLNR O43193 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7433172 0.92 CACNA1C (0.67) CACNA1CCACNA1FCACNA1DCACNA1SCYP1A2
SCHEMBL7431449 0.92 CACNA1C (0.78) CACNA1CCACNA1FCACNA1DCACNA1SCYP1A2
SCHEMBL7430572 0.91 CACNA1C (0.63) CACNA1CCACNA1FCACNA1DCACNA1SCYP1A2
SCHEMBL9765757 0.89 CACNA1C (0.69) CACNA1CCACNA1FCACNA1DCACNA1S
SCHEMBL11522396 0.88 CACNA1C (0.59) CACNA1CCACNA1FCACNA1DCACNA1SCYP1A2
SCHEMBL31579033 0.88 CACNA1C (0.73) CACNA1CCACNA1FCACNA1DCACNA1SCYP1A2
SCHEMBL7159720 0.87 CACNA1C (0.72) CACNA1CCACNA1FCACNA1DCACNA1SCYP1A2
SCHEMBL11012182 0.86 CACNA1C (0.65) CACNA1CCACNA1FCACNA1DCACNA1SCYP1A2
SCHEMBL11004883 0.85 CYP1A2 (0.71) CACNA1CCACNA1FCACNA1DCACNA1SCYP1A2
SCHEMBL10625412 0.85 CYP1A2 (0.71) CACNA1CCACNA1FCACNA1DCACNA1SCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4988717-A Optically active 1,4-dihydropyridine esters useful for treating circulatory illnesses BAYER AKTIENGESELLSCHAFT (DE) 1991-01-29 US disclosed
US-4849433-A The compound, (⃡)1,4-dihydro-2,6-dimethyl-4-(2'-nitrophenyl)-pyridine-3,5-dicarboxylic acid, methyl isobutyl ester, compositions containing same and a method for effecting coronary dilation BAYER AKTIENGESELLSCHAFT (DE) 1989-07-18 US disclosed
US-4703119-A Intermediates of optically active 1,4-dihydropyridines BAYER AKTIENGESELLSCHAFT (DE) 1987-10-27 US disclosed
US-4510310-A 1,4-Dihydro-2,6-dimethyl-4-(2'-chlorophenyl)-3,5-dicarboxylic acid,methyl or ethyl,trifluoroethyl ester BAYER AKTIENGESELLSCHAFT (DE) 1985-04-09 US disclosed