SCHEMBL9765706

SCHEMBL9765706

CC1=C(C(=O)OCc2ccccc2)C(c2ccccc2C#N)C(C(=O)OC(C)C)=C(C)N1

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NR3C2 P08235 3/20 0.51
GPBAR1 Q8TDU6 1/20 0.48
PDE1C Q14123 2/20 0.48
ADORA3 P0DMS8 1/20 0.47
KDM4E B2RXH2 3/20 0.46
MAPT P10636 2/20 0.46
TSHR P16473 2/20 0.46
ALDH1A1 P00352 1/20 0.46
GAA P10253 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
HSD17B10 Q99714 1/20 0.46
TDP1 Q9NUW8 1/20 0.45
CACNA1F O60840 1/20 0.44
CACNA1D Q01668 1/20 0.44
CACNA1S Q13698 1/20 0.44
CACNA1C Q13936 1/20 0.44
TP53 P04637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9765795 0.89 PDE1C (0.49) PDE1CADORA3KDM4EMAPTTSHR
SCHEMBL11742268 0.89 ADORA3 (0.55) PDE1CADORA3KDM4EMAPTTSHR
SCHEMBL11829322 0.89 NR3C2 (0.54) NR3C2ADORA3KDM4EMAPTTSHR
SCHEMBL6947811 0.87 CYP1A2 (0.56) NR3C2ADORA3KDM4EMAPTTSHR
SCHEMBL11823990 0.86 KDM4E (0.54) NR3C2KDM4EMAPTTSHRALDH1A1
SCHEMBL7163495 0.85 CACNA1C (0.58) NR3C2PDE1CADORA3KDM4EMAPT
SCHEMBL11695185 0.84 NR3C2 (0.48) NR3C2ADORA3KDM4EMAPTTSHR
SCHEMBL11366059 0.82 NR3C2 (0.39) NR3C2GPBAR1PDE1CADORA3KDM4E
SCHEMBL7158453 0.81 ADORA3 (0.55) ADORA3KDM4EMAPTTSHRALDH1A1
SCHEMBL11503470 0.80 ADORA3 (0.62) NR3C2PDE1CADORA3KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4988717-A Optically active 1,4-dihydropyridine esters useful for treating circulatory illnesses BAYER AKTIENGESELLSCHAFT (DE) 1991-01-29 US disclosed
US-4849433-A The compound, (⃡)1,4-dihydro-2,6-dimethyl-4-(2'-nitrophenyl)-pyridine-3,5-dicarboxylic acid, methyl isobutyl ester, compositions containing same and a method for effecting coronary dilation BAYER AKTIENGESELLSCHAFT (DE) 1989-07-18 US disclosed
US-4510310-A 1,4-Dihydro-2,6-dimethyl-4-(2'-chlorophenyl)-3,5-dicarboxylic acid,methyl or ethyl,trifluoroethyl ester BAYER AKTIENGESELLSCHAFT (DE) 1985-04-09 US disclosed