SCHEMBL9765795

SCHEMBL9765795

CC1=C(C(=O)O)C(c2ccccc2C#N)C(C(=O)OCc2ccccc2)=C(C)N1

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PDE1C Q14123 2/20 0.49
KDM4E B2RXH2 2/20 0.49
GAA P10253 2/20 0.49
TSHR P16473 2/20 0.49
HSD17B10 Q99714 2/20 0.49
ALDH1A1 P00352 1/20 0.49
MAPT P10636 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
CACNA1B Q00975 3/20 0.48
ADORA3 P0DMS8 1/20 0.47
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
GLA P06280 1/20 0.46
ADORA2B P29275 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11742268 0.93 ADORA3 (0.55) PDE1CKDM4EGAATSHRHSD17B10
SCHEMBL9765706 0.89 NR3C2 (0.51) PDE1CKDM4EGAATSHRHSD17B10
SCHEMBL6951436 0.87 KDM4E (0.46) PDE1CKDM4EGAAALDH1A1MAPT
SCHEMBL10642720 0.86 KDM4E (0.47) PDE1CKDM4EGAATSHRHSD17B10
SCHEMBL7164240 0.85 KDM4E (0.54) PDE1CKDM4EGAATSHRHSD17B10
SCHEMBL7158453 0.85 ADORA3 (0.55) KDM4EGAATSHRHSD17B10ALDH1A1
SCHEMBL7381384 0.83 ADORA3 (0.46) KDM4EGAATSHRHSD17B10ALDH1A1
Hydrochloric Acid SCHEMBL7380766 0.82 ADORA3 (0.46) KDM4EGAATSHRHSD17B10ALDH1A1
SCHEMBL7158466 0.81 ADORA3 (0.64) KDM4EGAATSHRHSD17B10ALDH1A1
SCHEMBL11859054 0.81 ADORA3 (0.51) KDM4EGAATSHRHSD17B10ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4988717-A Optically active 1,4-dihydropyridine esters useful for treating circulatory illnesses BAYER AKTIENGESELLSCHAFT (DE) 1991-01-29 US disclosed
US-4849433-A The compound, (⃡)1,4-dihydro-2,6-dimethyl-4-(2'-nitrophenyl)-pyridine-3,5-dicarboxylic acid, methyl isobutyl ester, compositions containing same and a method for effecting coronary dilation BAYER AKTIENGESELLSCHAFT (DE) 1989-07-18 US disclosed
US-4510310-A 1,4-Dihydro-2,6-dimethyl-4-(2'-chlorophenyl)-3,5-dicarboxylic acid,methyl or ethyl,trifluoroethyl ester BAYER AKTIENGESELLSCHAFT (DE) 1985-04-09 US disclosed