SCHEMBL9765722

SCHEMBL9765722

COC(=O)C1=C(C)NC(C)=C(C(=O)OCC(OC)c2ccccc2)C1c1ccccn1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.69
HSD17B10 Q99714 3/20 0.69
CASP1 P29466 3/20 0.64
CACNA1F O60840 6/20 0.54
CACNA1D Q01668 6/20 0.54
CACNA1S Q13698 6/20 0.54
CACNA1C Q13936 6/20 0.54
ALDH1A1 P00352 4/20 0.50
ADORA3 P0DMS8 2/20 0.50
CASP7 P55210 1/20 0.50
GAA P10253 1/20 0.49
HPGD P15428 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
ABCC4 O15439 1/20 0.46
NR1I2 O75469 1/20 0.46
ABCB11 O95342 1/20 0.46
LMNA P02545 1/20 0.46
NR3C1 P04150 1/20 0.46
CYP1A2 P05177 1/20 0.46
PGR P06401 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10763917 0.86 KDM4E (0.77) KDM4EHSD17B10CASP1CACNA1FCACNA1D
SCHEMBL7158896 0.84 KDM4E (0.90) KDM4EHSD17B10CASP1ALDH1A1ADORA3
SCHEMBL7160171 0.83 KDM4E (1.00) KDM4EHSD17B10CASP1CACNA1FCACNA1D
SCHEMBL10759503 0.81 KDM4E (0.77) KDM4EHSD17B10CASP1CACNA1FCACNA1D
SCHEMBL7160175 0.81 KDM4E (0.90) KDM4EHSD17B10CASP1CACNA1FCACNA1D
SCHEMBL10860930 0.81 KDM4E (0.79) KDM4EHSD17B10CASP1CACNA1FCACNA1D
SCHEMBL7158385 0.81 KDM4E (0.79) KDM4EHSD17B10CASP1ALDH1A1ADORA3
SCHEMBL9765691 0.80 ABCB11 (0.59) KDM4EHSD17B10CACNA1FCACNA1DCACNA1S
SCHEMBL7265761 0.80 KDM4E (0.70) KDM4EHSD17B10CASP1CACNA1FCACNA1D
SCHEMBL11824836 0.79 KDM4E (0.76) KDM4EHSD17B10CASP1CACNA1FCACNA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4988717-A Optically active 1,4-dihydropyridine esters useful for treating circulatory illnesses BAYER AKTIENGESELLSCHAFT (DE) 1991-01-29 US disclosed
US-4849433-A The compound, (⃡)1,4-dihydro-2,6-dimethyl-4-(2'-nitrophenyl)-pyridine-3,5-dicarboxylic acid, methyl isobutyl ester, compositions containing same and a method for effecting coronary dilation BAYER AKTIENGESELLSCHAFT (DE) 1989-07-18 US disclosed
US-4510310-A 1,4-Dihydro-2,6-dimethyl-4-(2'-chlorophenyl)-3,5-dicarboxylic acid,methyl or ethyl,trifluoroethyl ester BAYER AKTIENGESELLSCHAFT (DE) 1985-04-09 US disclosed