SCHEMBL9765691

SCHEMBL9765691

COC(=O)C1=C(C)NC(C)=C(C(=O)OCC(OC)c2ccccc2)C1c1ccccc1Cl

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB11 O95342 5/20 0.59
ADORA3 P0DMS8 5/20 0.59
CYP2C9 P11712 4/20 0.59
ADRA1A P35348 4/20 0.59
CYP1A2 P05177 4/20 0.59
CYP3A4 P08684 4/20 0.59
SCN5A Q14524 4/20 0.59
NR1I2 O75469 4/20 0.59
TBXA2R P21731 3/20 0.59
SLC6A3 Q01959 3/20 0.59
ABCB1 P08183 3/20 0.59
KDM4E B2RXH2 3/20 0.59
CYP2C19 P33261 3/20 0.59
KMT2A Q03164 3/20 0.59
HIF1A Q16665 3/20 0.59
HSD17B10 Q99714 3/20 0.59
LMNA P02545 3/20 0.59
SCN1A P35498 3/20 0.59
SCN2A Q99250 3/20 0.59
SCN3A Q9NY46 3/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14048599 0.83 CACNA1C (0.60) ABCB11ADORA3CYP2C9ADRA1ACYP1A2
SCHEMBL3031020 0.83 ADORA3 (0.82) ABCB11ADORA3CYP2C9ADRA1ACYP1A2
SCHEMBL29676073 0.83 KDM4E (0.68) ABCB11ADORA3CYP2C9ADRA1ACYP1A2
SCHEMBL3035724 0.83 KDM4E (0.68) ABCB11ADORA3CYP2C9ADRA1ACYP1A2
SCHEMBL6942341 0.81 CACNA1F (0.49) ABCB11ADORA3CYP2C9ADRA1ACYP1A2
SCHEMBL6942333 0.81 CACNA1F (0.49) ABCB11ADORA3CYP2C9ADRA1ACYP1A2
SCHEMBL3026759 0.81 KDM4E (0.62) ABCB11ADORA3CYP2C9ADRA1ACYP1A2
SCHEMBL9765722 0.80 KDM4E (0.69) ABCB11ADORA3ADRA1ACYP1A2SCN5A
SCHEMBL27421079 0.80 CYP2C9 (0.69) ABCB11ADORA3CYP2C9ADRA1ACYP1A2
SCHEMBL9485304 0.80 ABCB11 (0.72) ABCB11ADORA3CYP2C9ADRA1ACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4988717-A Optically active 1,4-dihydropyridine esters useful for treating circulatory illnesses BAYER AKTIENGESELLSCHAFT (DE) 1991-01-29 US disclosed
US-4849433-A The compound, (⃡)1,4-dihydro-2,6-dimethyl-4-(2'-nitrophenyl)-pyridine-3,5-dicarboxylic acid, methyl isobutyl ester, compositions containing same and a method for effecting coronary dilation BAYER AKTIENGESELLSCHAFT (DE) 1989-07-18 US disclosed
US-4510310-A 1,4-Dihydro-2,6-dimethyl-4-(2'-chlorophenyl)-3,5-dicarboxylic acid,methyl or ethyl,trifluoroethyl ester BAYER AKTIENGESELLSCHAFT (DE) 1985-04-09 US disclosed