SCHEMBL9765784

SCHEMBL9765784

CC1=C(C#N)C(c2ccccc2[N+](=O)[O-])C(C(=O)OC2CCCC2)=C(C)N1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.57
ADORA3 P0DMS8 3/20 0.57
LMNA P02545 3/20 0.57
CACNA1C Q13936 3/20 0.57
KDM4E B2RXH2 3/20 0.57
ABCC4 O15439 2/20 0.57
CACNA1F O60840 2/20 0.57
ABCB11 O95342 2/20 0.57
CYP1A2 P05177 2/20 0.57
ADORA2A P29274 2/20 0.57
ADORA1 P30542 2/20 0.57
OPRM1 P35372 2/20 0.57
SCN1A P35498 2/20 0.57
HTR2B P41595 2/20 0.57
CACNA1D Q01668 2/20 0.57
KCNH2 Q12809 2/20 0.57
CACNA1S Q13698 2/20 0.57
SCN5A Q14524 2/20 0.57
SCN2A Q99250 2/20 0.57
SCN3A Q9NY46 2/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9765793 0.86 ADORA3 (0.79) MAPTADORA3LMNACACNA1CKDM4E
SCHEMBL11357785 0.86 KDM4E (0.47) MAPTADORA3LMNACACNA1CKDM4E
SCHEMBL10693916 0.86 ADORA3 (0.78) MAPTADORA3LMNACACNA1CKDM4E
SCHEMBL10987755 0.84 CACNA1D (0.55) MAPTADORA3LMNACACNA1CKDM4E
SCHEMBL7265869 0.82 KDM4E (0.58) MAPTADORA3LMNACACNA1CKDM4E
SCHEMBL11746889 0.81 ADORA3 (0.59) MAPTADORA3LMNACACNA1CKDM4E
SCHEMBL204910 0.81 CUL4A (0.64) MAPTADORA3LMNACACNA1CKDM4E
SCHEMBL11737070 0.80 ADORA3 (0.58) MAPTADORA3LMNACACNA1CKDM4E
SCHEMBL10893501 0.78 NR3C2 (0.55) MAPTALDH1A1TP53NOTCH1NR3C2
SCHEMBL11521635 0.75 ADORA3 (0.47) MAPTADORA3LMNACACNA1CKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4988717-A Optically active 1,4-dihydropyridine esters useful for treating circulatory illnesses BAYER AKTIENGESELLSCHAFT (DE) 1991-01-29 US disclosed
US-4849433-A The compound, (⃡)1,4-dihydro-2,6-dimethyl-4-(2'-nitrophenyl)-pyridine-3,5-dicarboxylic acid, methyl isobutyl ester, compositions containing same and a method for effecting coronary dilation BAYER AKTIENGESELLSCHAFT (DE) 1989-07-18 US disclosed
US-4510310-A 1,4-Dihydro-2,6-dimethyl-4-(2'-chlorophenyl)-3,5-dicarboxylic acid,methyl or ethyl,trifluoroethyl ester BAYER AKTIENGESELLSCHAFT (DE) 1985-04-09 US disclosed