SCHEMBL9765807

SCHEMBL9765807

COC(=O)C1=C(C)NC(C)=C(C(=O)OC(C)C)C1c1ccnc2ccccc12

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 4/20 0.60
CACNA1C Q13936 4/20 0.60
ADORA3 P0DMS8 4/20 0.60
CYP3A4 P08684 3/20 0.60
CYP2C9 P11712 3/20 0.60
CYP2C19 P33261 3/20 0.60
ABCB11 O95342 3/20 0.60
KCNH2 Q12809 3/20 0.60
SCN5A Q14524 3/20 0.60
NR1I2 O75469 3/20 0.60
CYP2D6 P10635 2/20 0.60
KMT2A Q03164 2/20 0.60
NR3C1 P04150 2/20 0.60
PDE4D Q08499 2/20 0.60
PDE3A Q14432 2/20 0.60
MEN1 O00255 1/20 0.60
MLNR O43193 1/20 0.60
CYP2C8 P10632 1/20 0.60
ALOX15 P16050 1/20 0.60
TBXA2R P21731 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9401552 0.88 KDM4E (0.54) CYP1A2CACNA1CADORA3CYP3A4CYP2C9
SCHEMBL11826599 0.86 ADORA3 (0.60) CYP1A2CACNA1CADORA3CYP3A4CYP2C9
SCHEMBL11376558 0.83 NR3C2 (0.52) CYP1A2CACNA1CADORA3CYP3A4CYP2C9
SCHEMBL11365585 0.81 NR3C2 (0.42) CYP1A2CACNA1CADORA3CYP3A4CYP2C9
SCHEMBL9434406 0.81 KDM4E (0.58) CYP1A2CACNA1CADORA3CYP3A4CYP2C9
SCHEMBL11828335 0.80 KDM4E (0.51) CYP1A2CACNA1CADORA3CYP3A4CYP2C9
SCHEMBL11774395 0.80 SMN1; SMN2 (0.41) CYP1A2CACNA1CADORA3CYP3A4CYP2C9
SCHEMBL11525325 0.79 NR3C2 (0.50) CYP1A2CACNA1CADORA3CYP3A4CYP2C9
SCHEMBL7160381 0.78 KDM4E (0.83) CYP1A2CACNA1CADORA3CYP3A4CYP2C9
SCHEMBL11004140 0.77 CACNA1C (0.72) CYP1A2CACNA1CADORA3CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4988717-A Optically active 1,4-dihydropyridine esters useful for treating circulatory illnesses BAYER AKTIENGESELLSCHAFT (DE) 1991-01-29 US disclosed
US-4849433-A The compound, (⃡)1,4-dihydro-2,6-dimethyl-4-(2'-nitrophenyl)-pyridine-3,5-dicarboxylic acid, methyl isobutyl ester, compositions containing same and a method for effecting coronary dilation BAYER AKTIENGESELLSCHAFT (DE) 1989-07-18 US disclosed
US-4510310-A 1,4-Dihydro-2,6-dimethyl-4-(2'-chlorophenyl)-3,5-dicarboxylic acid,methyl or ethyl,trifluoroethyl ester BAYER AKTIENGESELLSCHAFT (DE) 1985-04-09 US disclosed