SCHEMBL9401552

SCHEMBL9401552

COC(=O)C1=C(C)NC(C)=C(C(=O)O)C1c1ccnc2ccccc12

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.54
HSD17B10 Q99714 5/20 0.54
PDE1C Q14123 1/20 0.54
CYP1A2 P05177 6/20 0.51
CYP3A4 P08684 5/20 0.51
CYP2C9 P11712 5/20 0.51
CYP2C19 P33261 5/20 0.51
ADORA3 P0DMS8 4/20 0.51
CACNA1C Q13936 4/20 0.51
MAPT P10636 4/20 0.51
KMT2A Q03164 4/20 0.51
ABCB11 O95342 3/20 0.51
KCNH2 Q12809 3/20 0.51
SCN5A Q14524 3/20 0.51
ALDH1A1 P00352 3/20 0.51
HPGD P15428 3/20 0.51
TSHR P16473 3/20 0.51
CYP2D6 P10635 3/20 0.51
CACNA1F O60840 3/20 0.51
CACNA1D Q01668 3/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11826599 0.89 ADORA3 (0.60) KDM4EHSD17B10PDE1CCYP1A2CYP3A4
SCHEMBL9765807 0.88 CYP1A2 (0.60) KDM4EHSD17B10PDE1CCYP1A2CYP3A4
SCHEMBL9434406 0.84 KDM4E (0.58) KDM4EHSD17B10PDE1CCYP1A2CYP3A4
SCHEMBL11525325 0.81 NR3C2 (0.50) KDM4EHSD17B10PDE1CCYP1A2CYP3A4
SCHEMBL9580965 0.81 CYP2C9 (0.48) KDM4EHSD17B10PDE1CCYP1A2CYP3A4
SCHEMBL9401663 0.81 KDM4E (0.58) KDM4EHSD17B10PDE1CCYP1A2CYP3A4
SCHEMBL7160175 0.77 KDM4E (0.90) KDM4EHSD17B10PDE1CCYP1A2CYP3A4
SCHEMBL9580964 0.76 CYP2C9 (0.51) KDM4EHSD17B10PDE1CCYP1A2CYP3A4
SCHEMBL6951320 0.76 ADORA3 (0.76) KDM4EHSD17B10PDE1CCYP1A2CYP3A4
SCHEMBL7414856 0.75 NR1I2 (0.67) KDM4EHSD17B10PDE1CCYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5286869-A Vasodilators and anticoagulants FUJIREBIO KABUSHIKI KAISHA (JP) 1994-02-15 US disclosed
EP-0403957-A2 Optical active 1,4-dihydropyridine derivates FUJIREBIO INC. (JP) 1990-12-27 EP disclosed