SCHEMBL9766006

SCHEMBL9766006

OC(CCCN1CCN(c2ncc(F)cn2)CC1)c1ccc(F)c2ccccc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 11/20 1.00
KDM4E B2RXH2 1/20 0.64
CYP1A2 P05177 1/20 0.64
GAA P10253 1/20 0.64
CYP2C9 P11712 1/20 0.64
DRD2 P14416 1/20 0.64
HTR1A P08908 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9766032 0.88 SIGMAR1 (0.98) SIGMAR1KDM4ECYP1A2GAACYP2C9
SCHEMBL13532633 0.82 SIGMAR1 (0.84) SIGMAR1KDM4ECYP1A2GAACYP2C9
SCHEMBL9766093 0.79 SIGMAR1 (0.73) SIGMAR1KDM4ECYP1A2GAACYP2C9
SCHEMBL9766068 0.79 SIGMAR1 (1.00) SIGMAR1KDM4ECYP1A2GAACYP2C9
Bmy-14802 SCHEMBL8457738 0.78 SIGMAR1 (1.00) SIGMAR1KDM4ECYP1A2GAACYP2C9
Bmy-14802 SCHEMBL467229 0.78 SIGMAR1 (1.00) SIGMAR1KDM4ECYP1A2GAACYP2C9
Ammonia Solution, Strong SCHEMBL9765999 0.78 SIGMAR1 (0.98) SIGMAR1KDM4ECYP1A2GAACYP2C9
SCHEMBL9766055 0.77 SIGMAR1 (0.64) SIGMAR1KDM4ECYP1A2GAACYP2C9
SCHEMBL13532647 0.77 SIGMAR1 (0.84) SIGMAR1KDM4ECYP1A2GAACYP2C9
Bmy-14802 SCHEMBL10843594 0.77 SIGMAR1 (0.97) SIGMAR1KDM4ECYP1A2GAACYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4994460-A Treatment or prevention of disorders resulting from central nervous system anoxia BRISTOL-MYERS SQUIBB CO. (US) 1991-02-19 US claimed
EP-0400661-A1 Agents for treatment of brain ischemia Bristol-Myers Squibb Company (US) 1990-12-05 EP claimed
US-4994460-A Treatment or prevention of disorders resulting from central nervous system anoxia BRISTOL-MYERS SQUIBB CO. (US) 1991-02-19 US disclosed
EP-0400661-A1 Agents for treatment of brain ischemia Bristol-Myers Squibb Company (US) 1990-12-05 EP disclosed