SCHEMBL9766076

SCHEMBL9766076

COC(=O)c1c(F)c(F)c(OC)c(F)c1F

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.52
MAPK1 P28482 1/20 0.52
SMN1; SMN2 Q16637 3/20 0.46
KMT2A Q03164 6/20 0.45
MEN1 O00255 5/20 0.45
CYP2C9 P11712 2/20 0.45
CYP1A2 P05177 1/20 0.45
KDM4E B2RXH2 2/20 0.41
GFER P55789 1/20 0.41
POLB P06746 1/20 0.41
MAPT P10636 2/20 0.41
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA7 P43166 1/20 0.40
CA9 Q16790 1/20 0.40
CA14 Q9ULX7 1/20 0.40
ALDH1A1 P00352 2/20 0.38
USP2 O75604 1/20 0.37
RECQL P46063 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27367262 0.96 TSHR (0.49) TSHRMAPK1SMN1; SMN2KMT2AMEN1
SCHEMBL8593844 0.93 TSHR (0.46) TSHRMAPK1SMN1; SMN2KMT2AMEN1
SCHEMBL9766080 0.91 TSHR (0.44) TSHRMAPK1SMN1; SMN2KMT2AMEN1
SCHEMBL522175 0.88 TSHR (0.61) TSHRMAPK1SMN1; SMN2KMT2AMEN1
SCHEMBL9766012 0.86 SMN1; SMN2 (0.46) TSHRMAPK1SMN1; SMN2KMT2AMEN1
SCHEMBL27326641 0.86 KDM4E (0.41) TSHRMAPK1SMN1; SMN2KMT2AMEN1
SCHEMBL8653304 0.86 KMT2A (0.50) TSHRMAPK1SMN1; SMN2KMT2AMEN1
SCHEMBL1719721 0.85 TSHR (0.59) TSHRMAPK1SMN1; SMN2KDM4EMAPT
SCHEMBL27388705 0.84 MEN1 (0.41) TSHRMAPK1SMN1; SMN2KMT2AMEN1
SCHEMBL27866508 0.84 TSHR (0.46) TSHRMAPK1SMN1; SMN2KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1064955-C Fluorine-containing benzoylguanidines MERCK PATENT GMBH (DE) 2001-04-25 CN disclosed
CN-1143632-A Fluorine-containing benzoylguanidines MERCK PATENT GMBH (DE) 1997-02-26 CN disclosed
EP-0266947-B1 HALOGENATED ESTERS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1991-12-04 EP disclosed
US-4853414-A 1-/2-ALKOXY-3,5-DIFLUOROBENZYL ESTERS OF 2,2-DIMETHYL-3-ALKYLCYCLOPROPIONIC ACID; INSECTICIDES; PESTICIDES IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1989-08-01 US disclosed
EP-0266947-A2 Halogenated esters IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1988-05-11 EP disclosed