SCHEMBL9766461

SCHEMBL9766461

COc1cc(N)c(Cl)cc1C(=O)NCCNC1CC1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 12/20 0.65
DRD2 P14416 3/20 0.63
HTR3A P46098 3/20 0.63
HTR3E A5X5Y0 2/20 0.63
HTR3B O95264 2/20 0.63
HTR3D Q70Z44 2/20 0.63
HTR3C Q8WXA8 2/20 0.63
CYP1A2 P05177 2/20 0.63
ADRA2A P08913 2/20 0.63
CYP2D6 P10635 2/20 0.63
ADRA2C P18825 2/20 0.63
DRD4 P21917 2/20 0.63
HTR2A P28223 2/20 0.63
HTR2C P28335 2/20 0.63
DRD3 P35462 2/20 0.63
HTR2B P41595 2/20 0.63
KCNH2 Q12809 2/20 0.63
SLC22A1 O15245 1/20 0.63
ALDH1A1 P00352 1/20 0.63
LMNA P02545 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15650737 0.85 HTR4 (0.83) HTR4DRD2HTR3ACYP1A2ADRA2A
SCHEMBL15651357 0.82 HTR4 (0.71) HTR4DRD2HTR3AHTR3EHTR3B
SCHEMBL22022238 0.82 HTR4 (0.71) HTR4DRD2HTR3AHTR3EHTR3B
SCHEMBL15650650 0.82 HTR4 (0.71) HTR4DRD2HTR3AHTR3EHTR3B
Monodeethylated-Mcp SCHEMBL15585981 0.81 HTR4 (0.70) HTR4DRD2HTR3AHTR3EHTR3B
SCHEMBL8041200 0.81 HTR4 (0.78) HTR4DRD4
SCHEMBL17069817 0.81 HTR4 (0.65) HTR4DRD2HTR3AHTR3EHTR3B
Hydrochloric Acid SCHEMBL7301566 0.81 RAB9A (0.67) HTR4DRD2HTR3AHTR3EHTR3B
SCHEMBL9766463 0.81 HTR4 (0.69) HTR4DRD2HTR3AHTR3EHTR3B
SCHEMBL15650947 0.80 HTR4 (0.68) HTR4DRD2HTR3AHTR3EHTR3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2022257-A None JP disclosed
US-5010108-A Treatment of gastrointestinal disorders POLI INDUSTRIA CHIMICA S.P.A. (IT) 1991-04-23 US disclosed
JP-H0222257-A N-CYCLOALKYLAMINOETHYLBENZAMIDE DERIVATIVE, ITS PRODUCTION AND PHARMACEUTICAL USE POLI IND CHIM SPA 1990-01-25 JP disclosed
EP-0333073-A2 N-cycloalkylaminoethylbenzamide derivatives, their synthesis and pharmaceutical preparations POLI INDUSTRIA CHIMICA S.p.A. (IT) 1989-09-20 EP disclosed