SCHEMBL9766631

SCHEMBL9766631

CCCCCCCCOc1ccc([C@H]2CC[C@H](C#Cc3ccc(F)nc3F)CC2)cc1.CCCCCOc1ccc([C@H]2CC[C@H](C#Cc3ccc(F)nc3F)CC2)cc1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 1/20 0.38
S1PR3 Q99500 1/20 0.37
HRH3 Q9Y5N1 3/20 0.36
CYP2C9 P11712 2/20 0.36
LMNA P02545 2/20 0.36
NR5A1 Q13285 1/20 0.35
LTA4H P09960 1/20 0.34
SPHK1 Q9NYA1 1/20 0.33
HTR1A P08908 1/20 0.33
DRD2 P14416 1/20 0.33
DRD1 P21728 1/20 0.33
DRD5 P21918 1/20 0.33
HTR2A P28223 1/20 0.33
DRD3 P35462 1/20 0.33
CRBN Q96SW2 1/20 0.33
CYP3A4 P08684 1/20 0.33
KCNH2 Q12809 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9158285 1.00 RAB9A (0.38) RAB9AS1PR3HRH3CYP2C9LMNA
SCHEMBL9158289 1.00 RAB9A (0.38) RAB9AS1PR3HRH3CYP2C9LMNA
SCHEMBL9157082 0.99 RAB9A (0.39) RAB9AS1PR3HRH3CYP2C9LMNA
SCHEMBL9157090 0.99 RAB9A (0.39) RAB9AS1PR3HRH3CYP2C9LMNA
SCHEMBL9160838 0.97 RAB9A (0.40) RAB9AHRH3CYP2C9LMNAHTR1A
SCHEMBL9160827 0.97 RAB9A (0.40) RAB9AHRH3CYP2C9LMNAHTR1A
SCHEMBL9766730 0.95 RAB9A (0.39) RAB9AHRH3CYP2C9LMNAHTR1A
SCHEMBL9766727 0.95 RAB9A (0.39) RAB9AHRH3CYP2C9LMNAHTR1A
SCHEMBL9160793 0.93 RAB9A (0.35) RAB9AHRH3CYP2C9HTR1ADRD2
SCHEMBL9160786 0.93 RAB9A (0.35) RAB9AHRH3CYP2C9HTR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0445248-A1 PYRIDINE DERIVATIVES. MERCK PATENT GMBH (DE) 1991-09-11 EP disclosed