SCHEMBL9766935

SCHEMBL9766935

CCCOC1=CC(=O)NC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.54
MAPT P10636 2/20 0.36
ALDH1A1 P00352 1/20 0.36
MAOA P21397 2/20 0.35
MAOB P27338 2/20 0.35
PIM1 P11309 1/20 0.34
PIM2 Q9P1W9 1/20 0.34
PDE4A P27815 2/20 0.33
GAA P10253 1/20 0.32
PDE7A Q13946 1/20 0.31
PDE7B Q9NP56 1/20 0.31
PDE4B Q07343 1/20 0.31
PDE4D Q08499 1/20 0.31
NAAA Q02083 1/20 0.31
ASAH1 Q13510 1/20 0.31
HSD17B10 Q99714 1/20 0.31
TSHR P16473 1/20 0.31
CA12 O43570 2/20 0.31
CA1 P00915 2/20 0.31
CA2 P00918 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9767275 0.90 HTT (0.53) HTTMAOAMAOBPDE4APDE4B
SCHEMBL9321078 0.89 HTT (0.51) HTTMAOAMAOBNAAATSHR
SCHEMBL9767396 0.87 HTT (0.50) HTTNAAATSHRLMNA
SCHEMBL9767026 0.87 HTT (0.50) HTTNAAATSHRLMNA
SCHEMBL9767272 0.87 HTT (0.50) HTTNAAATSHRLMNA
SCHEMBL9767347 0.78 HTT (0.53) HTT
SCHEMBL9767447 0.77 HTT (0.51) HTTMAPTALDH1A1PDE4APDE4B
SCHEMBL9767083 0.76 HTT (0.50) HTT
SCHEMBL9767015 0.73 HTT (0.51) HTTPDE4APDE4BPDE4DCA12
SCHEMBL9766990 0.69 HTT (0.43) HTTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5072006-A Chemical intermeidate; hypotensive agents, muscle relaxants RECHERCHE SYNTEX FRANCE S.A. (FR) 1991-12-10 US disclosed
US-4997846-A Smooth muscle relaxants, hypotensives RESEARCHE SYNTEX FRANCE, S.A. (FR) 1991-03-05 US disclosed
EP-0377966-A2 Novel benzopyranylpyrrolinone derivatives RECHERCHE SYNTEX FRANCE SA (FR) 1990-07-18 EP disclosed