SCHEMBL9768889

SCHEMBL9768889

O=C(c1ccncc1)C1COCOC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 4/20 0.44
KDM4E B2RXH2 2/20 0.44
POLB P06746 1/20 0.44
NAPRT Q6XQN6 1/20 0.42
NPC1 O15118 1/20 0.40
CYP1A2 P05177 2/20 0.40
CYP3A4 P08684 2/20 0.40
CYP2C9 P11712 1/20 0.40
ALDH1A1 P00352 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37
HTR2B P41595 1/20 0.37
MPO P05164 1/20 0.37
ADORA3 P0DMS8 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2A6 P11509 1/20 0.37
CYP2C19 P33261 1/20 0.37
CHRNB2 P17787 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9187512 0.81 MCL1 (0.44) NAPRTCYP1A2CYP2C9MEN1KMT2A
SCHEMBL9768803 0.80 ALDH1A1 (0.49) GAAKDM4EALDH1A1MEN1KMT2A
SCHEMBL6494263 0.78 KDM4E (0.58) GAAKDM4EPOLBNAPRTNPC1
SCHEMBL28957256 0.75 POLB (0.55) GAAKDM4EPOLBNAPRTNPC1
SCHEMBL9768794 0.74 NPC1 (0.34) KDM4ENAPRTNPC1CYP1A2CYP3A4
SCHEMBL9768828 0.74 POLB (0.39) GAAKDM4EPOLBNAPRTNPC1
SCHEMBL9768819 0.74 POLB (0.39) GAAKDM4EPOLBNAPRTNPC1
SCHEMBL11638730 0.73 SRD5A2 (0.58) GAAKDM4EPOLBNAPRTCYP1A2
SCHEMBL4672863 0.72 KDM4E (0.53) GAAKDM4EPOLBNAPRTCYP1A2
SCHEMBL4672867 0.70 MEN1 (0.62) GAAKDM4EPOLBNAPRTCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5023334-A Anthelmintic pyridinyl acylhydrazones THE UPJOHN COMPANY (US) 1991-06-11 US disclosed
US-5011932-A Anthelmintic pyridinyl acylhydrazones derivatives UPJOHN COMPANY (US) 1991-04-30 US disclosed
EP-0214158-A1 ANTHELMINTIC PYRIDINYL ACYLHYDRAZONES, METHOD OF USE AND COMPOSITIONS THE UPJOHN COMPANY (US) 1987-03-18 EP disclosed
WO-1986004582-A1 ANTHELMINTIC PYRIDINYL ACYLHYDRAZONES, METHOD OF USE AND COMPOSITIONS THE UPJOHN COMPANY (US) 1986-08-14 WO disclosed