SCHEMBL976923

SCHEMBL976923

O=C1C=C(c2ccccc2)CCC1c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DDB1 Q16531 1/20 0.47
CRBN Q96SW2 1/20 0.47
CFTR P13569 1/20 0.47
GOPC Q9HD26 1/20 0.47
CTRB1 P17538 1/20 0.41
CYP19A1 P11511 2/20 0.38
PDGFRA P16234 1/20 0.37
PRKACA P17612 1/20 0.37
KDR P35968 1/20 0.37
CDK8 P49336 1/20 0.37
CDK9 P50750 1/20 0.37
ROCK1 Q13464 1/20 0.37
CLK4 Q9HAZ1 1/20 0.37
DYRK1B Q9Y463 1/20 0.37
KMT2A Q03164 4/20 0.36
TSHR P16473 1/20 0.36
HCAR2 Q8TDS4 1/20 0.36
ALDH1A1 P00352 2/20 0.35
MEN1 O00255 2/20 0.35
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11548260 0.78 DDB1 (0.47) DDB1CRBNCFTRGOPCCTRB1
SCHEMBL12539690 0.73 CFTR (0.69) DDB1CRBNCFTRGOPCCTRB1
SCHEMBL13210441 0.71 DDB1 (0.57) DDB1CRBNCFTRGOPCCTRB1
SCHEMBL14880674 0.70 DDB1 (0.46) DDB1CRBNCFTRGOPCCTRB1
SCHEMBL9459051 0.69 TP53 (0.44) KMT2AMEN1TP53L3MBTL1NPC1
SCHEMBL27708579 0.68 DDB1 (0.53) DDB1CRBNCFTRGOPCCTRB1
SCHEMBL9469683 0.68 DDB1 (0.45) DDB1CRBNCFTRGOPCCTRB1
SCHEMBL24102958 0.67 DDB1 (0.43) DDB1CRBNCFTRGOPCCTRB1
SCHEMBL3534373 0.67 DDB1 (0.47) DDB1CRBNCFTRGOPCCTRB1
SCHEMBL11548049 0.67 DDB1 (0.47) DDB1CRBNCFTRGOPCCTRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7872029-B2 Chalcone and its analogs as agents for the inhibition of angiogenesis and related disease states BOWEN J PHILLIP 2011-01-18 US disclosed
US-20090018167-A1 Chalcone and its analogs as agents for the inhibition of angiogenesis and related disease states Robinson, Thomas Philip (US) 2009-01-15 US disclosed
US-20030027830-A1 Chalcone and its analogs as agents for the inhibition of angiogenesis and related disease states UNIVERSITY OF GEORGIA RESEARCH FOUNDATION, INC. 2003-02-06 US disclosed
US-20020040029-A1 Chalcone and its analogs as agents for the inhibition of angiogenesis and related disease states BOWEN, J. PHILLIP 2002-04-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020040029-A1 Chalcone and its analogs as agents for the inhibition of angiogenesis and related disease states FLT1, FLT4, VEGFA DDB1 4316/4885CRBN 951/4885CFTR 3754/4885
US-20090018167-A1 Chalcone and its analogs as agents for the inhibition of angiogenesis and related disease states FLT1, FLT4, VEGFA DDB1 4096/4885CRBN 952/4885CFTR 3262/4885
US-20030027830-A1 Chalcone and its analogs as agents for the inhibition of angiogenesis and related disease states FLT1, VEGFA, FLT4 DDB1 4254/4885CRBN 646/4885CFTR 3680/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.