SCHEMBL9769296

SCHEMBL9769296

O[C@@H](CNC1CC1)c1ccc2nnnn2c1

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 2/20 0.44
JAK2 O60674 3/20 0.39
JAK1 P23458 3/20 0.39
TYK2 P29597 3/20 0.39
JAK3 P52333 2/20 0.39
KDM4E B2RXH2 1/20 0.39
BCHE P06276 2/20 0.36
HRH1 P35367 1/20 0.34
HRH4 Q9H3N8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10584351 1.00 ADRB2 (0.44) ADRB2JAK2JAK1TYK2JAK3
SCHEMBL9769111 0.95 KDM4E (0.46) ADRB2JAK2JAK1TYK2JAK3
SCHEMBL9769104 0.95 KDM4E (0.46) ADRB2JAK2JAK1TYK2JAK3
SCHEMBL9769131 0.95 KDM4E (0.43) ADRB2JAK2JAK1TYK2JAK3
SCHEMBL9769140 0.95 KDM4E (0.43) ADRB2JAK2JAK1TYK2JAK3
SCHEMBL9769373 0.87 JAK2 (0.33) ADRB2JAK2JAK1TYK2JAK3
SCHEMBL9769377 0.87 JAK2 (0.33) ADRB2JAK2JAK1TYK2JAK3
SCHEMBL9769376 0.78 ADRB2 (0.46) ADRB2KDM4E
SCHEMBL9769372 0.78 ADRB2 (0.46) ADRB2KDM4E
SCHEMBL9769278 0.77 ADRB2 (0.43) ADRB2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5019578-A β-adrenergic agonists MERCK & CO., INC. (US) 1991-05-28 US disclosed
EP-0318092-A2 Novel beta-adrenergic agonists MERCK & CO. INC. (US) 1989-05-31 EP disclosed