SCHEMBL9772979

SCHEMBL9772979

COc1ccc2[nH]cc(CC(C)(C)NCC(O)c3ccc4nnnn4c3)c2c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 5/20 0.49
ADRB3 P13945 1/20 0.47
HTR2A P28223 3/20 0.40
MTNR1A P48039 4/20 0.40
GPR84 Q9NQS5 2/20 0.40
HTR2B P41595 3/20 0.39
MTNR1B P49286 2/20 0.39
HTR1A P08908 2/20 0.39
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 1/20 0.39
CYP1A1 P04798 1/20 0.39
MPO P05164 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
HPGD P15428 1/20 0.39
NQO2 P16083 1/20 0.39
RAB9A P51151 1/20 0.39
BLM P54132 1/20 0.39
PMP22 Q01453 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9772953 1.00 CYP2D6 (0.49) CYP2D6ADRB3HTR2AMTNR1AGPR84
SCHEMBL9773000 0.87 ADRB3 (0.59) CYP2D6ADRB3MEN1KMT2A
SCHEMBL9773011 0.87 ADRB3 (0.59) CYP2D6ADRB3MEN1KMT2A
SCHEMBL9773100 0.84 ADRB3 (0.52) CYP2D6ADRB3HTR2AGPR84HTR2B
SCHEMBL9773015 0.84 ADRB3 (0.52) CYP2D6ADRB3HTR2AGPR84HTR2B
SCHEMBL9773025 0.84 ADRB3 (0.52) CYP2D6ADRB3HTR2AGPR84HTR2B
SCHEMBL9773082 0.78 CYP2D6 (0.54) CYP2D6ADRB3HTR2AMTNR1AGPR84
SCHEMBL9773074 0.78 CYP2D6 (0.54) CYP2D6ADRB3HTR2AMTNR1AGPR84
Hydrochloric Acid SCHEMBL9773056 0.78 CYP2D6 (0.53) CYP2D6ADRB3HTR2AMTNR1AGPR84
Hydrochloric Acid SCHEMBL9773071 0.78 CYP2D6 (0.53) CYP2D6ADRB3HTR2AMTNR1AGPR84

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5030640-A Alpha-heterocyclic ethanolamino alkylindoles, growth promoters and feed efficiency agents for animals, bronchodilators, antidepressants, antiobesity agents MERCK & CO., INC. (US) 1991-07-09 US disclosed