Wr-190433

Wr-190433

SCHEMBL977482

O=C(C=Cc1ccccn1)c1ccccc1

nearest known ligand 0.66

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TUBB4A P04350 2/20 0.66
TUBB P07437 2/20 0.66
TUBA3C P0DPH7 2/20 0.66
TUBA1B P68363 2/20 0.66
TUBA4A P68366 2/20 0.66
TUBB4B P68371 2/20 0.66
TUBB3 Q13509 2/20 0.66
TUBB2A Q13885 2/20 0.66
TUBB8 Q3ZCM7 2/20 0.66
TUBA3E Q6PEY2 2/20 0.66
TUBA1A Q71U36 2/20 0.66
TUBA1C Q9BQE3 2/20 0.66
TUBB6 Q9BUF5 2/20 0.66
TUBB2B Q9BVA1 2/20 0.66
TUBB1 Q9H4B7 2/20 0.66
HSP90AA1 P07900 2/20 0.63
MAPT P10636 5/20 0.58
LMNA P02545 2/20 0.58
CYP1B1 Q16678 2/20 0.58
KEAP1 Q14145 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Wr-190433 SCHEMBL30880222 1.00 TUBB4A (0.66) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
Wr-190433 SCHEMBL29870441 1.00 TUBB4A (0.66) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
Wr-190433 SCHEMBL6180067 1.00 TUBB4A (0.66) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL15882450 0.94 TUBB4A (0.72) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL15882451 0.94 TUBB4A (0.72) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL11473136 0.91 TUBB4A (0.65) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL11473133 0.91 TUBB4A (0.65) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL28713225 0.88 TUBB4A (0.65) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL1604279 0.88 TUBB4A (0.65) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL9700985 0.86 TUBB4A (0.63) TUBB4ATUBBTUBA3CTUBA1BTUBA4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 27 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025235348-A1 MACHINE-LEARNED MODELS FOR PROCESSING STRUCTURAL REPRESENTATIONS OF THERAPEUTIC MATERIALS GOOGLE LLC (US) 2025-11-13 WO disclosed
WO-2020146636-A1 COMPOUNDS AND METHODS FOR TREATING OR PREVENTING HEART FAILURE DREXEL UNIVERSITY (US) 2020-07-16 WO disclosed
US-7872029-B2 Chalcone and its analogs as agents for the inhibition of angiogenesis and related disease states BOWEN J PHILLIP 2011-01-18 US disclosed
US-20090018167-A1 Chalcone and its analogs as agents for the inhibition of angiogenesis and related disease states Robinson, Thomas Philip (US) 2009-01-15 US disclosed
US-7432303-B2 Chalcone and its analogs as agents for the inhibition of angiogenesis and related disease states Bowen, J. Phillip (US) 2008-10-07 US disclosed
WO-2005121129-A1 NOVEL PROPENONE DERIVATIVES CONTAINING AROMATIC RINGS, A MAUFACTURING PROCESS THEREOF AND A COMPOSITION CONTAINING THE SAME USING AS AN ANTIINFLAMMATORY AGENT YEUNGNAM EDUCATIONAL FOUNDATION (KR) 2005-12-22 WO disclosed
US-20050148599-A1 Chalcone and its analogs as agents for the inhibition of angiogenesis and related disease states UNIVERSITY OF GEORGIA RESEARCH FOUNDATION, INC. 2005-07-07 US disclosed
US-6906105-B2 Chalcone and its analogs as agents for the inhibition of angiogenesis and related disease states BOWEN J PHILLIP (US) 2005-06-14 US disclosed
US-20050090532-A1 Medicinal uses of dihydropyrazoles THE PROCTER & GAMBLE COMPANY 2005-04-28 US disclosed
US-6878729-B2 Medicinal uses of dihydropyrazoles THE PROCTER & GAMBLE COMPANY (US) 2005-04-12 US disclosed
US-6462075-B1 USE OF CHALCONE AND ITS DERIVATIVES AS ANTITUMOR/ANTICANCER AGENTS AND TO TREAT A NUMBER OF CONDITIONS OR DISEASE STATES IN WHICH ANGIOGENESIS IS A FACTOR INCLUDING PSORIASIS, ACNE, ROSACEA, WARTS, ECZEMA, HEMANGIOMAS AND LYMPHANGIOGENESIS THE UNIVERSITY OF GEORGIA RESEARCH FOUNDATION, INC. 2002-10-08 US disclosed
US-20020040029-A1 Chalcone and its analogs as agents for the inhibition of angiogenesis and related disease states BOWEN, J. PHILLIP 2002-04-04 US disclosed
EP-0187711-B1 OCTAHYDROINDOLIZINE COMPOUNDS USEFUL AS ANALGESICS McNeilab, Inc. (US) 1990-08-29 EP disclosed
EP-0187711-A2 Octahydroindolizine compounds useful as analgesics McNeilab, Inc. (US) 1986-07-16 EP disclosed
US-4582836-A Octahydroindolizine compounds useful as analgesics MCNEILAB, INC. (US) 1986-04-15 US disclosed
US-4284829-A Hydroxyalkyl and oxoalkyl substituted phenols as analgesics and sedatives PFIZER INC. (US) 1981-08-18 US disclosed
US-4283569-A Hydroxyalkyl and oxoalkyl substituted phenols as analgesics and sedatives PFIZER INC. (US) 1981-08-11 US disclosed
US-4014889-A Process for preparing ketones BAYER AKTIENGESELLSCHAFT (DT) 1977-03-29 US disclosed
US-3991197-A ANALGESICS HOFFMANN-LA ROCHE INC. (US) 1976-11-09 US disclosed
US-3989708-A HYPOTENSIVE, CORONARY VESSEL DILATORS BAYER AKTIENGESELLSCHAFT (DT) 1976-11-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020040029-A1 Chalcone and its analogs as agents for the inhibition of angiogenesis and related disease states FLT1, FLT4, VEGFA TUBB4A 1158/4885TUBB 1335/4885TUBA3C 2006/4885
US-20090018167-A1 Chalcone and its analogs as agents for the inhibition of angiogenesis and related disease states FLT1, FLT4, VEGFA TUBB4A 1190/4885TUBB 1393/4885TUBA3C 2118/4885
US-20050090532-A1 Medicinal uses of dihydropyrazoles EPOR, VEGFA, FLT4 TUBB4A 136/4885TUBB 139/4885TUBA3C 332/4885
US-20050148599-A1 Chalcone and its analogs as agents for the inhibition of angiogenesis and related disease states FLT1, VEGFA, FLT4 TUBB4A 998/4885TUBB 947/4885TUBA3C 1706/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.