SCHEMBL9775863

SCHEMBL9775863

CNn1cc(C(=O)O)c(=O)c2cc3cc(F)c(N4CCNCC4)cc3nc21

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.52
LMNA P02545 6/20 0.52
KDM4E B2RXH2 6/20 0.52
HPGD P15428 5/20 0.52
HSD17B10 Q99714 5/20 0.52
BRD4 O60885 1/20 0.52
TSHR P16473 1/20 0.52
HTT P42858 1/20 0.52
CYP2J2 P51589 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52
CYP2C9 P11712 2/20 0.51
ATP6V1B2 P21281 1/20 0.51
TBXA2R P21731 1/20 0.51
EDNRA P25101 1/20 0.51
TARBP2 Q15633 1/20 0.51
TOP2A P11388 5/20 0.50
TOP2B Q02880 4/20 0.50
CYP1A2 P05177 1/20 0.50
DRD3 P35462 1/20 0.40
MEN1 O00255 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8941976 0.90 ALDH1A1 (0.45) ALDH1A1LMNAKDM4EHPGDHSD17B10
SCHEMBL9775907 0.90 ALDH1A1 (0.52) ALDH1A1LMNAKDM4EHPGDHSD17B10
SCHEMBL9775885 0.88 ALDH1A1 (0.47) ALDH1A1LMNAKDM4EHPGDHSD17B10
SCHEMBL9775945 0.87 ALDH1A1 (0.55) ALDH1A1LMNAKDM4EHPGDHSD17B10
Water SCHEMBL9785229 0.87 ALDH1A1 (0.54) ALDH1A1LMNAKDM4EHPGDHSD17B10
Water SCHEMBL9785232 0.87 ALDH1A1 (0.54) ALDH1A1LMNAKDM4EHPGDHSD17B10
SCHEMBL7240040 0.86 LMNA (0.51) ALDH1A1LMNAKDM4EHPGDHSD17B10
SCHEMBL8942031 0.85 KMT2A (0.46) ALDH1A1LMNAKDM4EHPGDHSD17B10
SCHEMBL8942041 0.85 TOP1 (0.42) ALDH1A1LMNAKDM4EHPGDHSD17B10
SCHEMBL9775916 0.85 ALDH1A1 (0.52) ALDH1A1LMNAKDM4EHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5004745-A Benzo[1,8]naphthyridine derivatives, their preparation and the compositions which contain them LABORATOIRE ROGER BELLON (FR) 1991-04-02 US disclosed
US-4990515-A Chemical intermediates RHONE-POULENC SANTE (FR) 1991-02-05 US disclosed
US-4970213-A Benzo(1,8)naphthyridine derivatives as intermediates RHONE-POULENC SANTE (FR) 1990-11-13 US disclosed