SCHEMBL9780272

SCHEMBL9780272

CCCc1c(OCCCSc2ccc(C(CCC(=O)O)Sc3ccc(C(=O)C(C)CC(=O)O)cc3)cc2)ccc(C(C)=O)c1O

nearest known ligand 0.65

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYSLTR2 Q9NS75 16/20 0.65
CYSLTR1 Q9Y271 16/20 0.65
PPARG P37231 2/20 0.47
PPARD Q03181 2/20 0.47
PPARA Q07869 2/20 0.47
GRM2 Q14416 1/20 0.47
LMNA P02545 1/20 0.45
CYP1A2 P05177 1/20 0.45
MAPT P10636 1/20 0.45
CYP2C9 P11712 1/20 0.45
NFKB1 P19838 1/20 0.45
BLM P54132 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9733858 0.90 CYSLTR2 (0.73) CYSLTR2CYSLTR1PPARGPPARDPPARA
SCHEMBL9780179 0.89 CYSLTR2 (0.62) CYSLTR2CYSLTR1PPARGPPARDPPARA
SCHEMBL9863237 0.89 CYSLTR2 (0.72) CYSLTR2CYSLTR1PPARGPPARDPPARA
Water SCHEMBL9780305 0.88 CYSLTR2 (0.71) CYSLTR2CYSLTR1PPARGPPARDPPARA
SCHEMBL9780365 0.84 CYSLTR2 (0.60) CYSLTR2CYSLTR1PPARGPPARDPPARA
SCHEMBL9733277 0.81 CYSLTR2 (0.73) CYSLTR2CYSLTR1PPARGPPARDPPARA
SCHEMBL9780238 0.81 CYSLTR2 (0.61) CYSLTR2CYSLTR1PPARGPPARDPPARA
SCHEMBL9780206 0.81 CYSLTR2 (0.59) CYSLTR2CYSLTR1PPARGPPARDPPARA
SCHEMBL10914002 0.80 CYSLTR2 (0.40) CYSLTR2CYSLTR1
SCHEMBL9780281 0.80 CYSLTR2 (0.82) CYSLTR2CYSLTR1PPARGPPARDPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0206741-B1 LEUKOTRIENE ANTAGONISTS MERCK FROSST CANADA INC. (CA) 1991-04-10 EP claimed
US-4990526-A Skin disorders, antiallergens, antiinflammatory agents MERCK FROSST CANADA, INC. (CA) 1991-02-05 US claimed
EP-0206741-A2 Leukotriene antagonists MERCK FROSST CANADA INC. (CA) 1986-12-30 EP claimed
US-4997926-A Viricides SCRIPPS CLINIC AND RESEARCH FOUNDATION (US) 1991-03-05 US disclosed
US-4990526-A Skin disorders, antiallergens, antiinflammatory agents MERCK FROSST CANADA, INC. (CA) 1991-02-05 US disclosed
EP-0206741-A2 Leukotriene antagonists MERCK FROSST CANADA INC. (CA) 1986-12-30 EP disclosed