SCHEMBL9780976

SCHEMBL9780976

COP(=O)(C#Cc1c(-c2ccc(F)cc2)c2ccccn2c1C(C)C)C[C@H](CC(=O)O)O[Si](c1ccccc1)(c1ccccc1)C(C)(C)C

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 3/20 0.31
SIRT6 Q8N6T7 2/20 0.31
ABCC3 O15438 1/20 0.31
ABCB11 O95342 1/20 0.31
HMGCR P04035 1/20 0.31
PGR P06401 1/20 0.31
ADORA3 P0DMS8 1/20 0.31
RXRA P19793 1/20 0.31
TBXA2R P21731 1/20 0.31
CCKAR P32238 1/20 0.31
ADRA1A P35348 1/20 0.31
PTGS2 P35354 1/20 0.31
NR4A2 P43354 1/20 0.31
PDE4D Q08499 1/20 0.31
SLC10A1 Q14973 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9853863 0.87 HMGCR (0.30) HMGCR
SCHEMBL9781040 0.87 HMGCR (0.30) HMGCR
SCHEMBL9655519 0.86 HMGCR (0.35) CYP2C9SIRT6ABCC3ABCB11HMGCR
SCHEMBL9695052 0.84 ABCB11 (0.39) CYP2C9SIRT6ABCC3ABCB11HMGCR
SCHEMBL9695065 0.84 ABCB11 (0.39) CYP2C9SIRT6ABCC3ABCB11HMGCR
SCHEMBL9696802 0.84 KCNK3 (0.31)
SCHEMBL9441753 0.82 ALDH1A1 (0.32) HMGCR
SCHEMBL8953003 0.82
SCHEMBL9780982 0.82
SCHEMBL9780988 0.82

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5025000-A Anticholesterol, antilipemic agents E. R. SQUIBB & SONS, INC. (US) 1991-06-18 US disclosed