SCHEMBL9781908

SCHEMBL9781908

[CH]=C(CC)c1ccc(OC)cc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 0.63
CA1 P00915 6/20 0.50
CA2 P00918 6/20 0.50
CES2 O00748 2/20 0.50
CES1 P23141 2/20 0.50
CA12 O43570 1/20 0.48
CA7 P43166 1/20 0.48
CA9 Q16790 1/20 0.48
CA14 Q9ULX7 1/20 0.48
KMT2A Q03164 1/20 0.47
GSK3B P49841 1/20 0.47
HDAC3 O15379 1/20 0.47
HDAC4 P56524 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC7 Q8WUI4 1/20 0.47
HDAC2 Q92769 1/20 0.47
HDAC10 Q969S8 1/20 0.47
HDAC11 Q96DB2 1/20 0.47
HDAC8 Q9BY41 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5694085 0.77 NR1I2 (0.68) NR1I2CA1CA2CES2CES1
SCHEMBL6232157 0.77 NR1I2 (1.00) NR1I2CA1CA2CES2CES1
SCHEMBL554922 0.77 NR1I2 (1.00) NR1I2CA1CA2CES2CES1
SCHEMBL554921 0.77 NR1I2 (1.00) NR1I2CA1CA2CES2CES1
SCHEMBL19974595 0.77 CES2 (0.58) NR1I2CA1CA2CES2CES1
SCHEMBL1866929 0.75 CA1 (0.60) NR1I2CA1CA2CES2CES1
SCHEMBL9782361 0.75 CES2 (0.56) NR1I2CA1CA2CES2CES1
SCHEMBL23252596 0.74 NR1I2 (0.63) NR1I2CA1CA2CES2CES1
SCHEMBL5085228 0.74 NR1I2 (0.63) NR1I2CA1CA2CES2CES1
SCHEMBL12973284 0.74 NR1I2 (0.63) NR1I2CA1CA2CES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4997836-A Inhibitor of platelet activating factor TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1991-03-05 US disclosed
EP-0368670-A1 Trisubstituted piperazine compounds, their production and use Takeda Chemical Industries, Ltd. (JP) 1990-05-16 EP disclosed
US-4474868-A ORGANIC PEROXIDE AND COMPOUND CONTAINING CATIONIC OXYGEN, SULFUR OXYGEN,SULFUR OR SELENIUM NIPPON OIL AND FATS CO., LTD. (JP) 1984-10-02 US disclosed