SCHEMBL9790063

SCHEMBL9790063

COC1CNCCC1NC(=O)c1cc(Cl)ccc1Oc1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 1/20 0.58
HTR4 Q13639 1/20 0.58
SLC6A2 P23975 5/20 0.44
SLC6A4 P31645 5/20 0.44
KCNH2 Q12809 5/20 0.44
LMNA P02545 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
SLC6A3 Q01959 2/20 0.42
STK39 Q9UEW8 2/20 0.41
CYP2D6 P10635 3/20 0.41
HTR2C P28335 6/20 0.41
HTR2B P41595 6/20 0.41
AHCY P23526 1/20 0.40
PTGER4 P35408 1/20 0.40
PARG Q86W56 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9790068 1.00 HTR3A (0.58) HTR3AHTR4SLC6A2SLC6A4KCNH2
SCHEMBL9790077 1.00 HTR3A (0.58) HTR3AHTR4SLC6A2SLC6A4KCNH2
SCHEMBL9532735 0.88 SLC6A2 (0.54) HTR3AHTR4SLC6A2SLC6A4KCNH2
SCHEMBL9790164 0.88 SLC6A2 (0.54) HTR3AHTR4SLC6A2SLC6A4KCNH2
SCHEMBL9790170 0.88 SLC6A2 (0.54) HTR3AHTR4SLC6A2SLC6A4KCNH2
SCHEMBL10122269 0.77 HTR3A (0.63) HTR3AHTR4
SCHEMBL10107504 0.77 HTR3A (0.63) HTR3AHTR4
SCHEMBL9721673 0.76 HTR3A (0.53) HTR3AHTR4
SCHEMBL9721683 0.76 HTR3A (0.53) HTR3AHTR4
SCHEMBL9721577 0.76 HTR3A (0.53) HTR3AHTR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4990521-A Treating diarhea JANSSEN PHARMACEUTICA (BE) 1991-02-05 US disclosed
EP-0251417-A2 4-(aroylamino) piperidinebutanamide derivatives JANSSEN PHARMACEUTICA N.V. (BE) 1988-01-07 EP disclosed