SCHEMBL9794843

SCHEMBL9794843

CCOC(=O)CC[C@H](NC(=O)c1ccc(OCCCc2c(N)nc(N)[nH]c2=O)cc1)C(=O)OCC

nearest known ligand 0.73

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GART P22102 17/20 0.73
ATIC P31939 2/20 0.56
DHFR P00374 1/20 0.51
FOLR2 P14207 1/20 0.50
FOLR1 P15328 1/20 0.50
SLC19A1 P41440 1/20 0.50
SLC46A1 Q96NT5 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9794846 1.00 GART (0.73) GARTATICDHFRFOLR2FOLR1
SCHEMBL9794852 0.88 GART (0.72) GARTATICFOLR2FOLR1SLC46A1
SCHEMBL9794858 0.88 GART (0.72) GARTATICFOLR2FOLR1SLC46A1
SCHEMBL9794911 0.84 GART (1.00) GARTATICFOLR2FOLR1SLC19A1
SCHEMBL10421274 0.80 GART (0.50) GARTATICDHFR
SCHEMBL10421275 0.80 GART (0.50) GARTATICDHFR
SCHEMBL7615333 0.80 GART (0.57) GARTDHFRFOLR2FOLR1SLC46A1
SCHEMBL9794864 0.80 GART (0.59) GARTATICDHFR
SCHEMBL7607120 0.79 GART (0.71) GARTATICFOLR1
SCHEMBL7609761 0.79 GART (0.70) GARTATICDHFRFOLR2FOLR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0409382-A1 Glutamic acid derivatives THE WELLCOME FOUNDATION LIMITED (GB) 1991-01-23 EP disclosed
US-4971973-A Antitumor agents from polyglutamic acid modified with n- 4- 3-(2,4-diamino-1,6-dihydro-6-oxo-5-pyrimidinyl!propoxyl!benzoyl -glutamic acid BURROUGHS WELLCOME CO. (US) 1990-11-20 US disclosed