SCHEMBL9794864

SCHEMBL9794864

CCOC(=O)c1ccc(OCCCc2c(N)nc(N)[nH]c2=O)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GART P22102 4/20 0.59
DHFR P00374 1/20 0.50
LMNA P02545 2/20 0.47
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
HSD17B10 Q99714 1/20 0.47
TBXAS1 P24557 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
ALDH1A1 P00352 2/20 0.45
MEN1 O00255 1/20 0.45
GAA P10253 1/20 0.45
KMT2A Q03164 1/20 0.45
MAPK1 P28482 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
MAOA P21397 1/20 0.44
KCNH2 Q12809 1/20 0.43
HRH3 Q9Y5N1 1/20 0.43
ATIC P31939 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9794867 0.86 GART (0.66) GARTDHFRALDH1A1KMT2AATIC
SCHEMBL9794872 0.85 GART (0.58) GARTLMNARAB9AALDH1A1MEN1
SCHEMBL9794846 0.80 GART (0.73) GARTDHFRATIC
SCHEMBL9794843 0.80 GART (0.73) GARTDHFRATIC
SCHEMBL9794911 0.74 GART (1.00) GARTATIC
SCHEMBL5166263 0.73 TDP1 (0.66) LMNATBXAS1TDP1L3MBTL1ALDH1A1
SCHEMBL6701399 0.73 TDP1 (0.74) LMNARAB9AHSD17B10TBXAS1TDP1
SCHEMBL9798438 0.72 L3MBTL1 (0.61) DHFRLMNATBXAS1TDP1L3MBTL1
Hydrochloric Acid SCHEMBL6983034 0.71 TDP1 (0.59) DHFRLMNATBXAS1TDP1L3MBTL1
SCHEMBL4247628 0.71 TDP1 (0.62) LMNATBXAS1TDP1L3MBTL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0409382-A1 Glutamic acid derivatives THE WELLCOME FOUNDATION LIMITED (GB) 1991-01-23 EP disclosed
WO-1990014340-A1 GLUTAMIC ACID DERIVATIVES THE WELLCOME FOUNDATION LIMITED (GB) 1990-11-29 WO disclosed
US-4971973-A Antitumor agents from polyglutamic acid modified with n- 4- 3-(2,4-diamino-1,6-dihydro-6-oxo-5-pyrimidinyl!propoxyl!benzoyl -glutamic acid BURROUGHS WELLCOME CO. (US) 1990-11-20 US disclosed