SCHEMBL9795472

SCHEMBL9795472

CC(C(=Cc1ccc(C#N)cc1)c1ccc(F)cc1)n1cncn1

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 18/20 0.47
CYP3A4 P08684 2/20 0.45
CYP2C19 P33261 2/20 0.45
CYP11B1 P15538 1/20 0.45
TSHR P16473 1/20 0.45
CYP11B2 P19099 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.39
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9795469 1.00 CYP19A1 (0.47) CYP19A1CYP3A4CYP2C19CYP11B1TSHR
Nitric Acid SCHEMBL9795315 0.79 RAB9A (0.40) CYP19A1CYP3A4SMN1; SMN2
Nitric Acid SCHEMBL9795307 0.79 RAB9A (0.40) CYP19A1CYP3A4SMN1; SMN2
SCHEMBL13285157 0.72 CYP19A1 (0.85) CYP19A1CYP3A4CYP2C19CYP11B1TSHR
SCHEMBL8104971 0.71 CYP19A1 (0.56) CYP19A1CYP3A4CYP2C19CYP11B1TSHR
SCHEMBL8104969 0.71 CYP19A1 (0.56) CYP19A1CYP3A4CYP2C19CYP11B1TSHR
SCHEMBL10361474 0.70 HSP90AA1 (0.49) CYP19A1CYP3A4CYP2C19CYP1A2CYP2C9
Hydrochloric Acid SCHEMBL9792757 0.69 HSP90AA1 (0.48) CYP19A1CYP3A4CYP2C19CYP1A2CYP2C9
SCHEMBL7709352 0.68 CYP19A1 (0.47) CYP19A1
SCHEMBL7709350 0.68 CYP19A1 (0.47) CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5032607-A Enzyme inhibitors IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1991-07-16 US disclosed
US-4866086-A PHENYLTRIAZOLYL OLEFINIC AROMATASE INHIBITORS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1989-09-12 US disclosed
EP-0299683-A2 Heterocyclic olefinic compounds and their use as aromatase inhibitors IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1989-01-18 EP disclosed