SCHEMBL9796263

SCHEMBL9796263

COc1ccc(N(C)C(C)=O)cc1C

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 3/20 0.49
NPC1 O15118 2/20 0.49
AHR P35869 1/20 0.49
ALDH1A1 P00352 6/20 0.46
LMNA P02545 1/20 0.46
HTT P42858 1/20 0.43
SMN1; SMN2 Q16637 4/20 0.41
RAB9A P51151 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.40
KMT2A Q03164 3/20 0.40
MEN1 O00255 2/20 0.40
TSHR P16473 2/20 0.40
TAS1R3 Q7RTX0 3/20 0.39
TAS1R1 Q7RTX1 3/20 0.39
TUBB1 Q9H4B7 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
PDK2 Q15119 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13503862 0.86 ALDH1A1 (0.48) POLBNPC1AHRALDH1A1LMNA
SCHEMBL19308888 0.79 MEN1 (0.51) POLBNPC1AHRALDH1A1HTT
SCHEMBL7094825 0.79 POLB (0.46) POLBNPC1AHRALDH1A1LMNA
SCHEMBL23034212 0.79 POLB (0.49) POLBNPC1AHRALDH1A1LMNA
SCHEMBL22537184 0.79 TAS1R3 (0.39) ALDH1A1KMT2AMEN1TSHRTAS1R3
SCHEMBL1911939 0.77 NQO2 (0.50) ALDH1A1LMNASMN1; SMN2KMT2AMEN1
SCHEMBL11198967 0.77 POLB (0.50) POLBNPC1AHRALDH1A1LMNA
SCHEMBL22537400 0.76 TAS1R3 (0.43) ALDH1A1SMN1; SMN2TAS1R3TAS1R1MAPT
SCHEMBL13503616 0.76 ALDH1A1 (0.43) POLBNPC1AHRALDH1A1LMNA
SCHEMBL850628 0.75 ALDH1A1 (0.46) POLBNPC1ALDH1A1LMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4997840-A Quinolone sulphonates having antihypertensive activity THE BOOTS COMPANY, PLC (GB) 1991-03-05 US disclosed
WO-1989007593-A1 THERAPEUTIC AGENTS THE BOOTS COMPANY PLC (GB) 1989-08-24 WO disclosed