SCHEMBL9797289

SCHEMBL9797289

CCCN1CCc2cc(OC)c(OC)cc2C(Oc2ccccc2)C1

nearest known ligand 0.51

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.51
CYP2D6 P10635 1/20 0.51
CHRNA7 P36544 2/20 0.47
MTNR1B P49286 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oxalic Acid SCHEMBL9806189 0.95 MTNR1B (0.48) CYP3A4CYP2D6CHRNA7MTNR1B
SCHEMBL9797437 0.91 CYP3A4 (0.50) CYP3A4CYP2D6CHRNA7MTNR1B
SCHEMBL9806155 0.89 MTNR1B (0.51) CYP3A4CYP2D6MTNR1B
SCHEMBL10416566 0.88 NR1I2 (0.45) CYP3A4CYP2D6
SCHEMBL9806154 0.88 GRIN1 (0.55) CYP3A4CYP2D6
Hydrochloric Acid SCHEMBL9806147 0.87 MAOA (0.44) CYP3A4CYP2D6
SCHEMBL9797731 0.84 CYP3A4 (0.67) CYP3A4CYP2D6CHRNA7
SCHEMBL9806164 0.84 ABCB1 (0.50) CYP3A4CYP2D6MTNR1B
Fumaric Acid SCHEMBL9797372 0.83 TRPV1 (0.47) CYP3A4CYP2D6MTNR1B
Maleic Acid SCHEMBL9797355 0.83 TRPV1 (0.47) CYP3A4CYP2D6MTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4988690-A Antidepressants HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1991-01-29 US claimed
US-4935418-A Medical compositions of 1-aryloxy-2,3,4,5-tetrahydro-3-benzazepines and use thereof HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1990-06-19 US claimed
US-4794181-A ANTIDEPRESSANTS, ANALGESICS HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1988-12-27 US claimed
US-5059688-A 1-aryloxy-2,3,4,5-tetrahydro-3-benzazepine preparation HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1991-10-22 US disclosed
US-4988690-A Antidepressants HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1991-01-29 US disclosed
US-4935418-A Medical compositions of 1-aryloxy-2,3,4,5-tetrahydro-3-benzazepines and use thereof HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1990-06-19 US disclosed
US-4794181-A ANTIDEPRESSANTS, ANALGESICS HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1988-12-27 US disclosed
EP-0096838-B1 1-ARYLOXY-2,3,4,5-TETRAHYDRO-3-BENZAZEPINES, A PROCESS FOR PREPARING THE SAME AND THEIR USE AS MEDICAMENTS HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1987-04-01 EP disclosed
EP-0096838-A1 1-Aryloxy-2,3,4,5-tetrahydro-3-benzazepines, a process for preparing the same and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1983-12-28 EP disclosed