SCHEMBL9799309

SCHEMBL9799309

CCCN(CCC)c1ccc(/C=C/c2ccc(/C=C/c3ccc([N+](=O)[O-])c([N+](=O)[O-])c3)nc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 10/20 0.49
MEN1 O00255 7/20 0.49
KMT2A Q03164 7/20 0.49
RAB9A P51151 4/20 0.49
NPC1 O15118 3/20 0.49
MAPK1 P28482 3/20 0.49
KDM4E B2RXH2 1/20 0.49
THRB P10828 1/20 0.49
ATM Q13315 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
ALDH3A1 P30838 2/20 0.47
LMNA P02545 5/20 0.40
ALDH1A1 P00352 2/20 0.40
GAA P10253 1/20 0.38
SMN1; SMN2 Q16637 3/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
HCAR3 P49019 1/20 0.36
POLB P06746 1/20 0.36
TDP1 Q9NUW8 2/20 0.36
CYP3A4 P08684 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9799316 1.00 MAPT (0.49) MAPTMEN1KMT2ARAB9ANPC1
SCHEMBL9799239 0.91 MAPT (0.51) MAPTMEN1KMT2ARAB9ANPC1
SCHEMBL9799245 0.91 MAPT (0.51) MAPTMEN1KMT2ARAB9ANPC1
SCHEMBL9799304 0.90 MAPT (0.47) MAPTMEN1KMT2ARAB9ANPC1
SCHEMBL9799299 0.90 MAPT (0.47) MAPTMEN1KMT2ARAB9ANPC1
SCHEMBL9798780 0.87 ALDH3A1 (0.52) MAPTMEN1KMT2ARAB9ANPC1
SCHEMBL9798784 0.87 ALDH3A1 (0.52) MAPTMEN1KMT2ARAB9ANPC1
SCHEMBL9799277 0.86 MAPT (0.49) MAPTMEN1KMT2ARAB9ANPC1
SCHEMBL9799284 0.86 MAPT (0.49) MAPTMEN1KMT2ARAB9ANPC1
SCHEMBL9798352 0.84 MAPT (0.41) MAPTMEN1KMT2ARAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0411103-A1 NON-LINEAR OPTICAL MATERIALS WITH VICINAL DONOR OR ACCEPTOR GROUPS MERCK PATENT GmbH (DE) 1991-02-06 EP disclosed
WO-1990009616-A1 NON-LINEAR OPTICAL MATERIALS WITH VICINAL DONOR OR ACCEPTOR GROUPS MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1990-08-23 WO disclosed