SCHEMBL9799511

SCHEMBL9799511

O=c1c2ccn(Cc3ccccc3)c2c2cccnc2n1C1CCCCC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 2/20 0.46
CNR1 P21554 6/20 0.44
CNR2 P34972 6/20 0.44
PDE4B Q07343 1/20 0.42
PDE4C Q08493 1/20 0.42
PDE4D Q08499 1/20 0.42
PDE3B Q13370 1/20 0.42
PDE3A Q14432 1/20 0.42
GAA P10253 1/20 0.42
ALOX15 P16050 1/20 0.42
DHPS P49366 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
ATM Q13315 1/20 0.40
TSHR P16473 1/20 0.40
CRHBP P24387 1/20 0.40
CRHR2 Q13324 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
GRM1 Q13255 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5872001 0.73 GAA (0.42) CNR1CNR2PDE4BPDE4DGAA
SCHEMBL1945900 0.66 SMN1; SMN2 (0.55) PDE4AMEN1KMT2ATSHRSMN1; SMN2
SCHEMBL1522680 0.66 DDB1 (0.42) PDE4BPDE4DGAAALOX15MEN1
SCHEMBL1522771 0.66 DDB1 (0.42) PDE4BPDE4DGAAALOX15MEN1
SCHEMBL7280534 0.65 PDE4A (0.83) PDE4APDE4BPDE4CPDE4DTSHR
SCHEMBL5871425 0.65 PDE4B (0.42) PDE4BPDE4DGAAALOX15MEN1
SCHEMBL1522541 0.64 DDB1 (0.43) PDE4BPDE4DGAAALOX15MEN1
SCHEMBL11871647 0.63 FEN1 (0.55) GAAALOX15MEN1KMT2AATM
SCHEMBL8696469 0.63 MGLL (0.41) GAAALOX15TSHRALDH1A1DDB1
SCHEMBL7272788 0.63 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4996212-A Antiinflammatory and anti-hyperproliferative compounds SCHERING CORPORATION (US) 1991-02-26 US claimed
US-4996212-A Antiinflammatory and anti-hyperproliferative compounds SCHERING CORPORATION (US) 1991-02-26 US disclosed
US-4859669-A Antiinflammatory and anti-hyperproliferative naphthyridin-4-ones SCHERING CORPORATION (US) 1989-08-22 US disclosed