SCHEMBL980

SCHEMBL980

Cc1[nH]cnc1CN1CCc2c(c3ccccc3n2C(C)C)C1=O

nearest known ligand 0.76

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.76
CYP1A2 P05177 1/20 0.76
CYP3A4 P08684 1/20 0.76
ADRA2C P18825 1/20 0.76
HTR2A P28223 1/20 0.76
HTR2C P28335 1/20 0.76
ADRA1A P35348 1/20 0.76
HTR2B P41595 1/20 0.76
HTR3A P46098 1/20 0.76
CASP6 P55212 1/20 0.75
CD44 P16070 1/20 0.41
DHFR P00374 1/20 0.37
FNTA P49354 1/20 0.37
FNTB P49356 1/20 0.37
PGGT1B P53609 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Maleic Acid SCHEMBL1533 0.93 KCNH2 (0.67) KCNH2CYP1A2CYP3A4ADRA2CHTR2A
Fumaric Acid SCHEMBL1534 0.93 KCNH2 (0.67) KCNH2CYP1A2CYP3A4ADRA2CHTR2A
SCHEMBL553 0.87 KCNH2 (0.69) KCNH2CYP1A2CYP3A4ADRA2CHTR2A
Alosetron SCHEMBL631 0.87 KCNH2 (1.00) KCNH2CYP1A2CYP3A4ADRA2CHTR2A
Alosetron SCHEMBL29377019 0.87 KCNH2 (1.00) KCNH2CYP1A2CYP3A4ADRA2CHTR2A
SCHEMBL20022665 0.86 HTR2A (0.56) KCNH2CYP1A2CYP3A4ADRA2CHTR2A
Alosetron SCHEMBL806 0.86 CASP6 (1.00) KCNH2CYP1A2CYP3A4ADRA2CHTR2A
Alosetron SCHEMBL29387635 0.86 CASP6 (1.00) KCNH2CYP1A2CYP3A4ADRA2CHTR2A
Alosetron SCHEMBL635233 0.85 KCNH2 (0.96) KCNH2CYP1A2CYP3A4ADRA2CHTR2A
SCHEMBL702 0.85 KCNH2 (0.78) KCNH2CYP1A2CYP3A4ADRA2CHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5360800-A Tetrahydro-1H-pyrido[4,3-b]indol-1-one derivatives GLAXO GROUP LIMITED (GB) 1994-11-01 US disclosed
US-5276050-A Administering for treatment of bulemia or seasonal affective disorder GLAXO GROUP LIMITED (GB) 1994-01-04 US disclosed
US-5225407-A Cognition activators GLAXO GROUP LIMITED (GB) 1993-07-06 US disclosed
EP-0450757-A2 Use of 5-hydroxytryptamine-antagonists in the treatment of mental disorders originating in childhood GLAXO GROUP LIMITED (GB) 1991-10-09 EP disclosed
EP-0411901-A2 Treatment of conditions involving excessive eating GLAXO GROUP LIMITED (GB) 1991-02-06 EP disclosed