SCHEMBL9802274

SCHEMBL9802274

c1ccc2c(c1)c1c3n2CCCC3CCC1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 6/20 0.59
KMT2A Q03164 6/20 0.59
HSD17B10 Q99714 5/20 0.59
ALDH1A1 P00352 4/20 0.59
HPGD P15428 1/20 0.59
SMPD1 P17405 1/20 0.47
MAPT P10636 5/20 0.44
TP53 P04637 3/20 0.44
MAPK1 P28482 3/20 0.44
LMNA P02545 2/20 0.44
CCR6 P51684 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
CYP1A2 P05177 2/20 0.43
CYP3A4 P08684 2/20 0.43
CYP2D6 P10635 2/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
KDM4E B2RXH2 5/20 0.40
GAA P10253 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12922443 0.79 KMT2A (0.68) MEN1KMT2AHSD17B10ALDH1A1MAPT
SCHEMBL19374171 0.76 ALDH1A1 (0.54) MEN1KMT2AHSD17B10ALDH1A1HPGD
SCHEMBL3174932 0.76 HSD17B10 (0.97) MEN1KMT2AHSD17B10ALDH1A1HPGD
SCHEMBL9802667 0.76 JAK3 (0.40) MEN1KMT2AHSD17B10ALDH1A1HPGD
SCHEMBL10836352 0.76 HSD17B10 (0.78) MEN1KMT2AHSD17B10ALDH1A1HPGD
SCHEMBL12922445 0.73 KMT2A (0.49) MEN1KMT2AHSD17B10ALDH1A1MAPT
SCHEMBL16433504 0.72 SMPD1 (0.46) MEN1KMT2AHSD17B10ALDH1A1SMPD1
SCHEMBL10992739 0.72 HSD17B10 (0.76) MEN1KMT2AHSD17B10ALDH1A1HPGD
SCHEMBL4152125 0.71 HTR1A (0.76) MEN1KMT2AHSD17B10ALDH1A1HPGD
SCHEMBL13925801 0.71 HSD17B10 (0.52) MEN1KMT2AHSD17B10ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5049563-A 5-hydroxytryptamine receptor antagonists DUPHAR INTERNATIONAL RESEARCH B.V. (NL) 1991-09-17 US disclosed
EP-0350129-A1 New annelated indoleketones with an imidazolylalkyl substituent DUPHAR INTERNATIONAL RESEARCH B.V (NL) 1990-01-10 EP disclosed