SCHEMBL9803101

SCHEMBL9803101

COC(=O)CC(=O)CC(O)/C=C/C1=C(c2ccc(F)cc2)C=C(c2ccccc2)C12CCCC2

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 4/20 0.34
ITGA4 P13612 4/20 0.34
ITGB7 P26010 4/20 0.34
NOS3 P29474 1/20 0.32
NOS1 P29475 1/20 0.32
NOS2 P35228 1/20 0.32
CA12 O43570 1/20 0.32
CA7 P43166 1/20 0.32
CA9 Q16790 1/20 0.32
CA14 Q9ULX7 1/20 0.32
NR4A2 P43354 2/20 0.32
PDE4D Q08499 2/20 0.32
NR1I2 O75469 1/20 0.32
ABCC3 O15438 1/20 0.32
ABCB11 O95342 1/20 0.32
HMGCR P04035 1/20 0.32
PGR P06401 1/20 0.32
ADORA3 P0DMS8 1/20 0.32
CYP2C9 P11712 1/20 0.32
RXRA P19793 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9802801 0.89 CYP2C9 (0.40) NR4A2PDE4DABCC3ABCB11HMGCR
SCHEMBL9803108 0.84 HMGCR (0.34) ITGB1ITGA4ITGB7NR4A2PDE4D
SCHEMBL9803360 0.82 HMGCR (0.47) NR4A2PDE4DNR1I2ABCC3ABCB11
SCHEMBL9803352 0.82 HMGCR (0.47) NR4A2PDE4DNR1I2ABCC3ABCB11
SCHEMBL9803192 0.80
SCHEMBL9616647 0.80
SCHEMBL9802811 0.80 HMGCR (0.36) NR4A2PDE4DABCC3ABCB11HMGCR
SCHEMBL9803466 0.72 TRPA1 (0.31) PGR
SCHEMBL9749704 0.72 PTGS2 (0.32) ITGB1ITGA4ITGB7HMGCRPTGS2
SCHEMBL9749709 0.72 PTGS2 (0.32) ITGB1ITGA4ITGB7HMGCRPTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5001128-A HMG-COA reductase inhibitors RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1991-03-19 US disclosed
WO-1990010444-A1 NOVEL HMG-CoA REDUCTASE INHIBITORS RORER INTERNATIONAL (HOLDINGS), INC. (US) 1990-09-20 WO disclosed
US-4904691-A Novel HMG-CoA reductase inhibitors RORER PHARMACEUTICAL CORPORATION (US) 1990-02-27 US disclosed