SCHEMBL9803233

SCHEMBL9803233

Cc1cc(=O)[nH]c2c1C(=O)CC(C)(C)C2

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.44
MAPK1 P28482 2/20 0.43
BRD4 O60885 2/20 0.43
BUB1 O43683 10/20 0.41
HSD17B10 Q99714 1/20 0.41
MEN1 O00255 1/20 0.40
ALPL P05186 1/20 0.40
KMT2A Q03164 1/20 0.40
ALDH1A1 P00352 1/20 0.40
TSHR P16473 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1220108 0.75 HSD17B10 (0.42) HTTMAPK1BRD4BUB1HSD17B10
SCHEMBL5004730 0.73 MAPK1 (0.54) MAPK1BRD4BUB1HSD17B10MEN1
SCHEMBL9802765 0.71 PTK2 (0.47) MAPK1BRD4BUB1HSD17B10ALDH1A1
SCHEMBL12820867 0.69 HSD17B10 (0.41) MAPK1BRD4BUB1HSD17B10MEN1
SCHEMBL12820992 0.69 HSD17B10 (0.41) MAPK1BRD4BUB1HSD17B10MEN1
SCHEMBL10796689 0.68 HTT (0.46) HTTMAPK1BRD4HSD17B10MEN1
SCHEMBL4325559 0.68 CYP2C19 (0.45) HTTBRD4BUB1HSD17B10ALPL
SCHEMBL370336 0.68 TDP1 (0.46) HTTMAPK1BRD4HSD17B10MEN1
SCHEMBL14896164 0.68 BUB1 (0.44) MAPK1BUB1ALPL
SCHEMBL14896227 0.67 ALPL (0.49) HTTBUB1ALPLALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5068334-A Analgesics and antipyretics KARL THOMAE GMBH (DE) 1991-11-26 US disclosed
EP-0338228-A2 Use of quinoline-2,5-diones in a medicament having an analgesic, antipyretic and/or antiphlogistic activity Dr. Karl Thomae GmbH (DE) 1989-10-25 EP disclosed