SCHEMBL9804254

SCHEMBL9804254

CCOc1c(F)cc(C(=CC=Cc2ccc(F)c(Oc3ccccc3)c2)C(F)(F)F)cc1F

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TUBB1 Q9H4B7 2/20 0.37
MAPT P10636 4/20 0.35
NPC1 O15118 3/20 0.35
RAB9A P51151 3/20 0.35
KMT2A Q03164 4/20 0.33
MEN1 O00255 3/20 0.33
KDM4E B2RXH2 3/20 0.33
LMNA P02545 2/20 0.33
GAA P10253 1/20 0.33
ALDH1A1 P00352 2/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
RELA Q04206 1/20 0.32
TNFRSF1A P19438 1/20 0.32
PKM P14618 1/20 0.32
RXRA P19793 1/20 0.32
PPARG P37231 1/20 0.32
LTA4H P09960 1/20 0.32
CYP1A1 P04798 1/20 0.31
CYP1B1 Q16678 1/20 0.31
MAPK1 P28482 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9804250 1.00 TUBB1 (0.37) TUBB1MAPTNPC1RAB9AKMT2A
SCHEMBL9804355 0.90 RELA (0.40) TUBB1MAPTNPC1RAB9AKMT2A
SCHEMBL9804361 0.90 RELA (0.40) TUBB1MAPTNPC1RAB9AKMT2A
SCHEMBL9494665 0.81 PARP10 (0.36) NPC1RAB9AKMT2AMEN1GAA
SCHEMBL9494663 0.81 PARP10 (0.36) NPC1RAB9AKMT2AMEN1GAA
SCHEMBL9804643 0.75 TLR4 (0.38) NPC1RAB9AKMT2AMEN1
SCHEMBL9804647 0.75 TLR4 (0.38) NPC1RAB9AKMT2AMEN1
SCHEMBL9491929 0.75 PARP10 (0.34) NPC1RAB9AKMT2AMEN1GAA
SCHEMBL9491927 0.75 PARP10 (0.34) NPC1RAB9AKMT2AMEN1GAA
SCHEMBL9804536 0.73 RELA (0.39) MAPTNPC1RAB9AKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0240121-B1 DIPHENYL ETHER DERIVATIVES IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1991-04-17 EP disclosed
EP-0390228-A2 Chemical intermediates IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1990-10-03 EP disclosed
US-4791139-A Diphenyl ether derivatives and their use as insecticides IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1988-12-13 US disclosed
EP-0240121-A2 Diphenyl ether derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1987-10-07 EP disclosed