SCHEMBL9804528

SCHEMBL9804528

CC(=O)OCCCCN(C)c1ccc(C=Cc2ccncc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.47
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47
MAPT P10636 2/20 0.47
MEN1 O00255 1/20 0.47
ALOX15 P16050 1/20 0.47
CASP1 P29466 1/20 0.47
HBB P68871 1/20 0.47
KMT2A Q03164 1/20 0.47
SNCA P37840 1/20 0.40
HDAC1 Q13547 2/20 0.40
KDM1A O60341 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
HPGD P15428 2/20 0.37
CYP1A2 P05177 2/20 0.37
CYP2D6 P10635 2/20 0.37
RAD52 P43351 1/20 0.37
KDM4E B2RXH2 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9804507 0.89 SMN1; SMN2 (0.43) SMN1; SMN2NPC1RAB9AMAPTMEN1
SCHEMBL10613260 0.85 MAPK1 (0.42) SMN1; SMN2NPC1RAB9AMAPTMEN1
SCHEMBL3038631 0.82 CYP2A6 (0.41) SMN1; SMN2KMT2ARAD52LMNAALDH1A1
SCHEMBL9804522 0.80 SMN1; SMN2 (0.56) SMN1; SMN2NPC1RAB9AMAPTMEN1
SCHEMBL10613289 0.80 SMN1; SMN2 (0.56) SMN1; SMN2NPC1RAB9AMAPTMEN1
SCHEMBL9804533 0.77 MAPT (0.56) SMN1; SMN2NPC1RAB9AMAPTMEN1
SCHEMBL9804751 0.77 RAD52 (0.46) MAPTMEN1KMT2AHPGDCYP1A2
SCHEMBL9804650 0.77 RAD52 (0.51) RAD52KDM4EBCHECHRM2CHRM4
SCHEMBL18774386 0.77 MAPT (0.59) SMN1; SMN2NPC1RAB9AMAPTMEN1
SCHEMBL20764316 0.76 ALDH1A1 (0.46) NPC1RAB9AMAPTCYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0290591-B1 MATERIALS WITH NITROGENOUS SIX-MEMBERED RINGS MERCK PATENT GmbH (DE) 1991-03-13 EP disclosed
EP-0290591-A1 MATERIALS WITH NITROGENOUS SIX-MEMBERED RINGS. MERCK PATENT GMBH (DE) 1988-11-17 EP disclosed
WO-1988004305-A1 MATERIALS WITH NITROGENOUS SIX-MEMBERED RINGS MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1988-06-16 WO disclosed