SCHEMBL9804718

SCHEMBL9804718

N#CC(CCc1ccccc1C(F)(F)F)(Cc1cnccn1)c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PIEZO1 Q92508 2/20 0.40
VNN1 O95497 1/20 0.33
NR3C2 P08235 1/20 0.32
LNPEP Q9UIQ6 1/20 0.32
SGMS2 Q8NHU3 1/20 0.32
HPSE Q9Y251 1/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2B Q13224 1/20 0.32
MAOA P21397 1/20 0.32
MAOB P27338 1/20 0.32
IDO1 P14902 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
KCNN4 O15554 1/20 0.30
TRPV1 Q8NER1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9804741 0.83 CYP19A1 (0.34) NR3C2HPSEMAOBIDO1TDP1
SCHEMBL9804823 0.82 EBP (0.39) VNN1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL9804889 0.78 CYP1A2 (0.37) VNN1GRIN1GRIN2BCYP1A2CYP3A4
SCHEMBL10405109 0.78 CYP3A4 (0.40) CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL9804794 0.77 CYP19A1 (0.37) CYP1A2CYP2C9CYP2C19
SCHEMBL9804838 0.75 VNN1 (0.38) PIEZO1VNN1NR3C2GRIN1GRIN2B
SCHEMBL9557183 0.73 HSP90AA1 (0.44) CYP3A4CYP2C9CYP2C19
SCHEMBL9804735 0.72 CYP19A1 (0.42) VNN1GRIN1GRIN2B
SCHEMBL9804667 0.70 CYP19A1 (0.40) CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL9804805 0.70 CYP19A1 (0.40) CYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0276920-B1 (2-CYANO-2-(PHENYL OR NAPHTHYL)-2-SUBSTITUTED-ETHYL) PYRAZINES, PYRIMIDINES AND PYRIDAZINES ROHM AND HAAS COMPANY (US) 1991-04-03 EP claimed
EP-0276920-B1 (2-CYANO-2-(PHENYL OR NAPHTHYL)-2-SUBSTITUTED-ETHYL) PYRAZINES, PYRIMIDINES AND PYRIDAZINES ROHM AND HAAS COMPANY (US) 1991-04-03 EP disclosed