SCHEMBL9804838

SCHEMBL9804838

N#CC(CCc1cccc(C(F)(F)F)c1)(Cc1cnccn1)c1ccccc1Cl

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
VNN1 O95497 1/20 0.38
GAA P10253 1/20 0.38
CTSC P53634 5/20 0.37
GRIN2B Q13224 4/20 0.37
GRIN1 Q05586 3/20 0.37
TAAR1 Q96RJ0 1/20 0.36
MIF P14174 1/20 0.35
NR3C2 P08235 1/20 0.34
P4HB P07237 1/20 0.34
MRGPRX4 Q96LA9 1/20 0.34
MAOB P27338 1/20 0.34
PIEZO1 Q92508 1/20 0.34
KDM4E B2RXH2 1/20 0.34
POLB P06746 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9804762 0.87 CTSC (0.39) VNN1CTSCGRIN2BGRIN1TAAR1
SCHEMBL9804841 0.82 CYP3A4 (0.38) KDM4EPOLB
SCHEMBL9804735 0.82 CYP19A1 (0.42) VNN1GAACTSCGRIN2BGRIN1
SCHEMBL9557231 0.78 CYP19A1 (0.39) TAAR1MIFMAOBKDM4E
SCHEMBL9804823 0.77 EBP (0.39) VNN1
SCHEMBL9804718 0.75 PIEZO1 (0.40) VNN1GRIN2BGRIN1NR3C2MAOB
SCHEMBL9804794 0.74 CYP19A1 (0.37) KDM4E
SCHEMBL9804916 0.73 CYP19A1 (0.38) VNN1GAAGRIN2BGRIN1KDM4E
SCHEMBL9557665 0.72 TAAR1 (0.48) GAAGRIN2BGRIN1TAAR1MIF
SCHEMBL10371526 0.72 CYP19A1 (0.46) VNN1CTSCGRIN2BTAAR1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0276920-B1 (2-CYANO-2-(PHENYL OR NAPHTHYL)-2-SUBSTITUTED-ETHYL) PYRAZINES, PYRIMIDINES AND PYRIDAZINES ROHM AND HAAS COMPANY (US) 1991-04-03 EP disclosed
EP-0276920-A1 (2-Cyano-2-(phenyl or naphthyl)-2-substituted-ethyl) pyrazines, pyrimidines and pyridazines ROHM AND HAAS COMPANY (US) 1988-08-03 EP disclosed