SCHEMBL9804757

SCHEMBL9804757

CCCCC(C#N)(Cc1cnccn1)c1cccc2ccccc12

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TLR7 Q9NYK1 1/20 0.36
CNR2 P34972 4/20 0.34
CNR1 P21554 3/20 0.34
HTR1B P28222 2/20 0.33
ALOX15 P16050 4/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
HTR1D P28221 1/20 0.32
GBA1 P04062 1/20 0.31
KDM4E B2RXH2 2/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
EBP Q15125 1/20 0.31
SIGMAR1 Q99720 1/20 0.31
HRH1 P35367 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9804684 0.83 EBP (0.33) CNR2CNR1HTR1BALOX15HTR1D
SCHEMBL11662606 0.80 ADRA2A (0.43) HTR1BALOX15HTR1DEBPSIGMAR1
SCHEMBL9804675 0.77 CYP2C9 (0.39) TLR7CNR2CNR1GBA1EBP
SCHEMBL11469880 0.76 POLB (0.43) KDM4EL3MBTL1
SCHEMBL9804764 0.74 KMT2A (0.40) SMN1; SMN2KDM4E
SCHEMBL9804851 0.74 KDM4E (0.36) SMN1; SMN2KDM4EL3MBTL1
SCHEMBL9804810 0.74 CYP19A1 (0.39) SMN1; SMN2KDM4EL3MBTL1EBPSIGMAR1
SCHEMBL9804889 0.70 CYP1A2 (0.37) TLR7KDM4EEBPSIGMAR1HRH1
SCHEMBL28039400 0.68 HTR1B (0.39) CNR2CNR1HTR1BSMN1; SMN2HTR1D
SCHEMBL10371965 0.68 CYP1A2 (0.39) SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0276920-B1 (2-CYANO-2-(PHENYL OR NAPHTHYL)-2-SUBSTITUTED-ETHYL) PYRAZINES, PYRIMIDINES AND PYRIDAZINES ROHM AND HAAS COMPANY (US) 1991-04-03 EP disclosed
EP-0276920-A1 (2-Cyano-2-(phenyl or naphthyl)-2-substituted-ethyl) pyrazines, pyrimidines and pyridazines ROHM AND HAAS COMPANY (US) 1988-08-03 EP disclosed