SCHEMBL9806943

SCHEMBL9806943

CCCCOCCOC(=O)C1=C(N)NC(C)=C(C(=O)OCCCN2CCC(c3ccccc3)(c3ccccc3)CC2)C1c1cccc([N+](=O)[O-])c1

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 8/20 0.75
ADRA1D P25100 7/20 0.75
ADRA1B P35368 7/20 0.75
ADRA2A P08913 6/20 0.75
ADRA2B P18089 6/20 0.75
ADRA2C P18825 6/20 0.75
ADORA3 P0DMS8 3/20 0.75
TDP1 Q9NUW8 3/20 0.75
ABCB1 P08183 2/20 0.75
MAPT P10636 2/20 0.75
MEN1 O00255 1/20 0.75
TP53 P04637 1/20 0.75
CYP1A2 P05177 1/20 0.75
CHRM2 P08172 1/20 0.75
CYP3A4 P08684 1/20 0.75
HTR1A P08908 1/20 0.75
CHRM5 P08912 1/20 0.75
CYP2D6 P10635 1/20 0.75
CYP2C9 P11712 1/20 0.75
DRD2 P14416 1/20 0.75

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9806881 0.96 ADRA1A (0.70) ADRA1AADRA1DADRA1BADRA2AADRA2B
SCHEMBL10744249 0.96 ADRA1A (0.82) ADRA1AADRA1DADRA1BADRA2AADRA2B
SCHEMBL9806968 0.94 ADRA1A (0.78) ADRA1AADRA1DADRA1BADRA2AADRA2B
SCHEMBL9806899 0.93 ADRA1A (0.82) ADRA1AADRA1DADRA1BADRA2AADRA2B
SCHEMBL10759010 0.92 ADRA1A (0.76) ADRA1AADRA1DADRA1BADRA2AADRA2B
SCHEMBL9806930 0.92 ADRA1A (0.83) ADRA1AADRA1DADRA1BADRA2AADRA2B
SCHEMBL9806964 0.91 ADRA1A (0.74) ADRA1AADRA1DADRA1BADRA2AADRA2B
SCHEMBL9807024 0.91 ADRA1A (0.83) ADRA1AADRA1DADRA1BADRA2AADRA2B
SCHEMBL9807029 0.91 ADRA1A (0.83) ADRA1AADRA1DADRA1BADRA2AADRA2B
SCHEMBL9806895 0.89 ADRA1A (0.78) ADRA1AADRA1DADRA1BADRA2AADRA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5064839-A Vasodilators, coronary disorders, hypotensive BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1991-11-12 US disclosed